1WOF
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![BU of 1wof by Molmil](/molmil-images/mine/1wof) | Crystal Structure Of SARS-CoV Mpro in Complex with an Inhibitor N1 | 分子名称: | 3C-like proteinase, N-[(5-METHYLISOXAZOL-3-YL)CARBONYL]-L-ALANYL-L-VALYL-N~1~-((1S)-4-ETHOXY-4-OXO-1-{[(3S)-2-OXOPYRROLIDIN-3-YL]METHYL}BUT-2-ENYL)-L-LEUCINAMIDE | 著者 | Yang, H, Bartlam, M, Xue, X, Yang, K, Liang, W, Rao, Z. | 登録日 | 2004-08-18 | 公開日 | 2005-08-30 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Design of Wide-Spectrum Inhibitors Targeting Coronavirus Main Proteases. Plos Biol., 3, 2005
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7JXY
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![BU of 7jxy by Molmil](/molmil-images/mine/7jxy) | Structure of TTBK1 kinase domain in complex with Compound 18 | 分子名称: | (3S)-1-[1-(2-aminopyrimidin-4-yl)-1H-pyrazolo[4,3-c]pyridin-6-yl]-3-methylpent-1-yn-3-ol, Tau-tubulin kinase 1 | 著者 | Chodaprambil, J.V. | 登録日 | 2020-08-28 | 公開日 | 2021-05-19 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | Discovery of Potent and Brain-Penetrant Tau Tubulin Kinase 1 (TTBK1) Inhibitors that Lower Tau Phosphorylation In Vivo. J.Med.Chem., 64, 2021
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7JXX
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![BU of 7jxx by Molmil](/molmil-images/mine/7jxx) | Structure of TTBK1 kinase domain in complex with Compound 3 | 分子名称: | 4-(2-amino-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-11-yl)-2-methylbut-3-yn-2-ol, SODIUM ION, Tau-tubulin kinase 1 | 著者 | Chodaprambil, J.V. | 登録日 | 2020-08-28 | 公開日 | 2021-05-19 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.56 Å) | 主引用文献 | Discovery of Potent and Brain-Penetrant Tau Tubulin Kinase 1 (TTBK1) Inhibitors that Lower Tau Phosphorylation In Vivo. J.Med.Chem., 64, 2021
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2TPR
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![BU of 2tpr by Molmil](/molmil-images/mine/2tpr) | |
1F6M
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![BU of 1f6m by Molmil](/molmil-images/mine/1f6m) | CRYSTAL STRUCTURE OF A COMPLEX BETWEEN THIOREDOXIN REDUCTASE, THIOREDOXIN, AND THE NADP+ ANALOG, AADP+ | 分子名称: | 3-AMINOPYRIDINE-ADENINE DINUCLEOTIDE PHOSPHATE, FLAVIN-ADENINE DINUCLEOTIDE, THIOREDOXIN 1, ... | 著者 | Lennon, B.W, Williams Jr, C.H, Ludwig, M.L. | 登録日 | 2000-06-22 | 公開日 | 2000-08-30 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.95 Å) | 主引用文献 | Twists in catalysis: alternating conformations of Escherichia coli thioredoxin reductase. Science, 289, 2000
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