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4HRA
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Crystal Structure of DOT1L in Complex with EPZ-5676
分子名称: 5'-[{cis-3-[2-(5-tert-butyl-1H-benzimidazol-2-yl)ethyl]cyclobutyl}(propan-2-yl)amino]-5'-deoxyadenosine, Histone-lysine N-methyltransferase, H3 lysine-79 specific, ...
著者Jin, L.
登録日2012-10-26
公開日2013-07-31
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (3.15 Å)
主引用文献Potent inhibition of DOT1L as treatment of MLL-fusion leukemia.
Blood, 122, 2013
<12

 

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件を2024-10-02に公開中

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