3TB0
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![BU of 3tb0 by Molmil](/molmil-images/mine/3tb0) | |
3TAY
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5KV9
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![BU of 5kv9 by Molmil](/molmil-images/mine/5kv9) | Crystal structure of a hPIV haemagglutinin-neuraminidase-inhibitor complex | 分子名称: | 1,2-ETHANEDIOL, 2,6-anhydro-3,4,5-trideoxy-5-[(2-methylpropanoyl)amino]-4-(4-phenyl-1H-1,2,3-triazol-1-yl)-D-glycero-D-galacto-non-2-en onic acid, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Dirr, L, El-Deeb, I.M, Chavas, L.M.G, Guillon, P, von Itzstein, M. | 登録日 | 2016-07-13 | 公開日 | 2017-07-12 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | The impact of the butterfly effect on human parainfluenza virus haemagglutinin-neuraminidase inhibitor design. Sci Rep, 7, 2017
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3EWI
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![BU of 3ewi by Molmil](/molmil-images/mine/3ewi) | Structural analysis of the C-terminal domain of murine CMP-Sialic acid Synthetase | 分子名称: | N-acylneuraminate cytidylyltransferase | 著者 | Oschlies, M, Dickmanns, A, Stummeyer, K, Gerardy-Schahn, R, Ficner, R, Muenster-Kuehnel, A.K. | 登録日 | 2008-10-15 | 公開日 | 2009-08-18 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | A C-terminal phosphatase module conserved in vertebrate CMP-sialic acid synthetases provides a tetramerization interface for the physiologically active enzyme. J.Mol.Biol., 393, 2009
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5KV8
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![BU of 5kv8 by Molmil](/molmil-images/mine/5kv8) | Crystal structure of a hPIV haemagglutinin-neuraminidase-inhibitor complex | 分子名称: | 1,2-ETHANEDIOL, 2,6-anhydro-3,4,5-trideoxy-4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]-5-[(2-methylpropanoyl)amino]-D-glycero-D-galacto -non-2-enonic acid, 2-acetamido-2-deoxy-alpha-D-glucopyranose, ... | 著者 | Dirr, L, El-Deeb, I.M, Chavas, L.M.G, Guillon, P, von Itzstein, M. | 登録日 | 2016-07-13 | 公開日 | 2017-07-12 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.949 Å) | 主引用文献 | The impact of the butterfly effect on human parainfluenza virus haemagglutinin-neuraminidase inhibitor design. Sci Rep, 7, 2017
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8V9A
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![BU of 8v9a by Molmil](/molmil-images/mine/8v9a) | GII.NA1 Loreto 1257 norovirus protruding domain | 分子名称: | 1,2-ETHANEDIOL, Capsid protein VP1 | 著者 | Kher, G, Kim, I, Pancera, M, Hansman, G. | 登録日 | 2023-12-07 | 公開日 | 2024-06-19 | 最終更新日 | 2024-07-31 | 実験手法 | X-RAY DIFFRACTION (1.67 Å) | 主引用文献 | Development of a broad-spectrum therapeutic Fc-nanobody for human noroviruses. J.Virol., 98, 2024
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8V96
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![BU of 8v96 by Molmil](/molmil-images/mine/8v96) | GII.14 M7 norovirus protruding domain | 分子名称: | 1,2-ETHANEDIOL, Capsid protein VP1 | 著者 | Kher, G, Prewitt, A, Pancera, M, Hansman, G. | 登録日 | 2023-12-07 | 公開日 | 2024-06-19 | 最終更新日 | 2024-07-31 | 実験手法 | X-RAY DIFFRACTION (1.44 Å) | 主引用文献 | Development of a broad-spectrum therapeutic Fc-nanobody for human noroviruses. J.Virol., 98, 2024
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8V98
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![BU of 8v98 by Molmil](/molmil-images/mine/8v98) | GII.24 Loreto 1972 norovirus protruding domain | 分子名称: | 1,2-ETHANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, Capsid protein VP1 | 著者 | Kher, G, Prewitt, A, Pancera, M, Hansman, G. | 登録日 | 2023-12-07 | 公開日 | 2024-06-19 | 最終更新日 | 2024-07-31 | 実験手法 | X-RAY DIFFRACTION (1.74 Å) | 主引用文献 | Development of a broad-spectrum therapeutic Fc-nanobody for human noroviruses. J.Virol., 98, 2024
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8V95
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![BU of 8v95 by Molmil](/molmil-images/mine/8v95) | GII.8 Amsterdam norovirus protruding domain | 分子名称: | 1,2-ETHANEDIOL, Capsid protein (Fragment) | 著者 | Kher, G, Prewitt, A, Pancera, M, Hansman, G. | 登録日 | 2023-12-07 | 公開日 | 2024-06-19 | 最終更新日 | 2024-07-31 | 実験手法 | X-RAY DIFFRACTION (1.73 Å) | 主引用文献 | Development of a broad-spectrum therapeutic Fc-nanobody for human noroviruses. J.Virol., 98, 2024
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8V99
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![BU of 8v99 by Molmil](/molmil-images/mine/8v99) | GII.26 Leon 4509 norovirus protruding domain | 分子名称: | 1,2-ETHANEDIOL, ACETATE ION, Capsid protein VP1, ... | 著者 | Kher, G, Reese, T, Pancera, M, Hansman, G. | 登録日 | 2023-12-07 | 公開日 | 2024-06-19 | 最終更新日 | 2024-07-31 | 実験手法 | X-RAY DIFFRACTION (1.47 Å) | 主引用文献 | Development of a broad-spectrum therapeutic Fc-nanobody for human noroviruses. J.Virol., 98, 2024
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8V97
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![BU of 8v97 by Molmil](/molmil-images/mine/8v97) | GII.17 CS-E1 norovirus protruding domain | 分子名称: | 1,2-ETHANEDIOL, Capsid protein VP1, DI(HYDROXYETHYL)ETHER | 著者 | Kher, G, Prewitt, A, Pancera, M, Hansman, G. | 登録日 | 2023-12-07 | 公開日 | 2024-06-19 | 最終更新日 | 2024-07-31 | 実験手法 | X-RAY DIFFRACTION (1.27 Å) | 主引用文献 | Development of a broad-spectrum therapeutic Fc-nanobody for human noroviruses. J.Virol., 98, 2024
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2DWR
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8EN4
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![BU of 8en4 by Molmil](/molmil-images/mine/8en4) | Structure of GII.4 norovirus in complex with Nanobody 53 | 分子名称: | 1,2-ETHANEDIOL, Nanobody 53, VP1 | 著者 | Kher, G, Sabin, C, Koromyslova, A, Pancera, M, Hansman, G. | 登録日 | 2022-09-28 | 公開日 | 2023-03-15 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Direct Blockade of the Norovirus Histo-Blood Group Antigen Binding Pocket by Nanobodies. J.Virol., 97, 2023
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8EN5
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![BU of 8en5 by Molmil](/molmil-images/mine/8en5) | Structure of GII.4 norovirus in complex with Nanobody 56 | 分子名称: | 1,2-ETHANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, GII.4 P domain, ... | 著者 | Kher, G, Sabin, C, Pancera, M, Koromyslova, A, Hansman, G. | 登録日 | 2022-09-28 | 公開日 | 2023-03-15 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Direct Blockade of the Norovirus Histo-Blood Group Antigen Binding Pocket by Nanobodies. J.Virol., 97, 2023
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8EN0
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![BU of 8en0 by Molmil](/molmil-images/mine/8en0) | Structure of GII.17 norovirus in complex with Nanobody 7 | 分子名称: | Capsid protein VP1, Nanobody 7 | 著者 | Kher, G, Sabin, C, Koromyslova, A, Pancera, M, Hansman, G. | 登録日 | 2022-09-28 | 公開日 | 2023-03-15 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.99 Å) | 主引用文献 | Direct Blockade of the Norovirus Histo-Blood Group Antigen Binding Pocket by Nanobodies. J.Virol., 97, 2023
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8EMZ
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![BU of 8emz by Molmil](/molmil-images/mine/8emz) | Structure of GII.17 norovirus in complex with Nanobody 2 | 分子名称: | 1,2-ETHANEDIOL, GII.17 P domain, Nanobody 2 | 著者 | Kher, G, Sabin, C, Pancera, M, Koromyslova, A, Hansman, G. | 登録日 | 2022-09-28 | 公開日 | 2023-03-15 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Direct Blockade of the Norovirus Histo-Blood Group Antigen Binding Pocket by Nanobodies. J.Virol., 97, 2023
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8EN1
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![BU of 8en1 by Molmil](/molmil-images/mine/8en1) | Structure of GII.4 norovirus in complex with Nanobody 30 | 分子名称: | GII.4 P domain, Nanobody 30 | 著者 | Kher, G, Sabin, C, Pancera, M, Koromyslova, A, Hansman, G. | 登録日 | 2022-09-28 | 公開日 | 2023-03-15 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Direct Blockade of the Norovirus Histo-Blood Group Antigen Binding Pocket by Nanobodies. J.Virol., 97, 2023
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8EN6
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![BU of 8en6 by Molmil](/molmil-images/mine/8en6) | Structure of GII.4 norovirus in complex with Nanobody 76 | 分子名称: | 1,2-ETHANEDIOL, DIMETHYL SULFOXIDE, GII.4 P domain, ... | 著者 | Kher, G, Sabin, C, Pancera, M, Koromyslova, A, Hansman, G. | 登録日 | 2022-09-28 | 公開日 | 2023-03-15 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Direct Blockade of the Norovirus Histo-Blood Group Antigen Binding Pocket by Nanobodies. J.Virol., 97, 2023
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8EMY
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![BU of 8emy by Molmil](/molmil-images/mine/8emy) | Structure of GII.4 norovirus in complex with Nanobody 82 | 分子名称: | 1,2-ETHANEDIOL, GII.4 P domain, Nanobody 82 | 著者 | Kher, G, Sabin, C, Pancera, M, Koromyslova, A, Hansman, G. | 登録日 | 2022-09-28 | 公開日 | 2023-03-15 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Direct Blockade of the Norovirus Histo-Blood Group Antigen Binding Pocket by Nanobodies. J.Virol., 97, 2023
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8EN2
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![BU of 8en2 by Molmil](/molmil-images/mine/8en2) | Structure of GII.10 norovirus in complex with Nanobody 34 | 分子名称: | 1,2-ETHANEDIOL, GII.10 P domain, Nanobody 34 | 著者 | Kher, G, Sabin, C, Koromyslova, A, Pancera, M, Hansman, G. | 登録日 | 2022-09-28 | 公開日 | 2023-03-15 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Direct Blockade of the Norovirus Histo-Blood Group Antigen Binding Pocket by Nanobodies. J.Virol., 97, 2023
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8EN3
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![BU of 8en3 by Molmil](/molmil-images/mine/8en3) | Structure of GII.17 norovirus in complex with Nanobody 45 | 分子名称: | 1,2-ETHANEDIOL, Capsid protein VP1, Nanobody 45 | 著者 | Kher, G, Sabin, C, Pancera, M, Koromyslova, A, Hansman, G. | 登録日 | 2022-09-28 | 公開日 | 2023-03-15 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Direct Blockade of the Norovirus Histo-Blood Group Antigen Binding Pocket by Nanobodies. J.Virol., 97, 2023
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7SEA
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![BU of 7sea by Molmil](/molmil-images/mine/7sea) | Crystal structure of human Fibrillarin in complex with compound 2 from cocktail soak | 分子名称: | 6-(trifluoromethyl)pyrimidin-4-amine, DIMETHYL SULFOXIDE, FORMIC ACID, ... | 著者 | Shi, Y, El-Deeb, I.M, Masic, V, Hartley-Tassell, L, Maggioni, A, von Itzstein, M, Ve, T. | 登録日 | 2021-09-30 | 公開日 | 2022-02-09 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.91 Å) | 主引用文献 | Discovery of Cofactor Competitive Inhibitors against the Human Methyltransferase Fibrillarin. Pharmaceuticals, 15, 2021
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7SE7
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![BU of 7se7 by Molmil](/molmil-images/mine/7se7) | Crystal structure of human Fibrillarin in complex with S-adenosyl-L-methionine | 分子名称: | S-ADENOSYLMETHIONINE, rRNA 2'-O-methyltransferase fibrillarin | 著者 | Shi, Y, El-Deeb, I.M, Masic, V, Hartley-Tassell, L, Maggioni, A, von Itzstein, M, Ve, T. | 登録日 | 2021-09-30 | 公開日 | 2022-02-09 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Discovery of Cofactor Competitive Inhibitors against the Human Methyltransferase Fibrillarin. Pharmaceuticals, 15, 2021
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7SED
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![BU of 7sed by Molmil](/molmil-images/mine/7sed) | Crystal structure of human Fibrillarin in complex with compound 2a | 分子名称: | FORMIC ACID, N-(piperidin-4-yl)-6-(trifluoromethyl)pyrimidin-4-amine, rRNA 2'-O-methyltransferase fibrillarin | 著者 | Shi, Y, El-Deeb, I.M, Masic, V, Hartley-Tassell, L, Maggioni, A, von Itzstein, M, Ve, T. | 登録日 | 2021-09-30 | 公開日 | 2022-02-09 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Discovery of Cofactor Competitive Inhibitors against the Human Methyltransferase Fibrillarin. Pharmaceuticals, 15, 2021
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7SEC
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![BU of 7sec by Molmil](/molmil-images/mine/7sec) | Crystal structure of human Fibrillarin in complex with compound 1a | 分子名称: | 2-[(8S)-4-oxo-2-(trifluoromethyl)-4,5-dihydropyrazolo[1,5-a]pyrazin-6-yl]acetamide, DIMETHYL SULFOXIDE, FORMIC ACID, ... | 著者 | Shi, Y, El-Deeb, I.M, Masic, V, Hartley-Tassell, L, Maggioni, A, von Itzstein, M, Ve, T. | 登録日 | 2021-09-30 | 公開日 | 2022-02-09 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Discovery of Cofactor Competitive Inhibitors against the Human Methyltransferase Fibrillarin. Pharmaceuticals, 15, 2021
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