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1YJD
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BU of 1yjd by Molmil
Crystal structure of human CD28 in complex with the Fab fragment of a mitogenic antibody (5.11A1)
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Fab fragment of 5.11A1 antibody heavy chain, Fab fragment of 5.11A1 antibody light chain, ...
著者Evans, E.J, Esnouf, R.M, Manso-Sancho, R, Gilbert, R.J.C, James, J.R, Sorensen, P, Stuart, D.I, Davis, S.J.
登録日2005-01-14
公開日2005-02-15
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Crystal structure of a soluble CD28-Fab complex
Nat.Immunol., 6, 2005
6EON
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BU of 6eon by Molmil
Galactanase BT0290
分子名称: Beta-galactosidase, CALCIUM ION, alpha-D-galactopyranose
著者Basle, A, Munoz, J, Gilbert, H.
登録日2017-10-10
公開日2017-11-29
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献A surface endogalactanase in Bacteroides thetaiotaomicron confers keystone status for arabinogalactan degradation.
Nat Microbiol, 3, 2018
6EUI
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BU of 6eui by Molmil
The GH43, Beta 1,3 Galactosidase, BT3683 with galactose
分子名称: Beta-glucanase, CALCIUM ION, beta-D-galactopyranose
著者Cartmell, A, Gilbert, H.J.
登録日2017-10-30
公開日2018-10-17
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (1.76 Å)
主引用文献A surface endogalactanase in Bacteroides thetaiotaomicron confers keystone status for arabinogalactan degradation.
Nat Microbiol, 3, 2018
6EUJ
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BU of 6euj by Molmil
The GH43, Beta 1,3 Galactosidase, BT0265
分子名称: Beta-glucanase
著者Cartmell, A, Gilbert, H.J.
登録日2017-10-30
公開日2018-10-17
最終更新日2019-10-16
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献A surface endogalactanase in Bacteroides thetaiotaomicron confers keystone status for arabinogalactan degradation.
Nat Microbiol, 3, 2018
6EUF
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BU of 6euf by Molmil
The GH43, Beta 1,3 Galactosidase, BT0265
分子名称: Beta-glucanase, alpha-L-arabinofuranose-(1-3)-[alpha-L-arabinofuranose-(1-4)][beta-D-glucopyranuronic acid-(1-6)]beta-D-galactopyranose-(1-6)-beta-D-galactopyranose, alpha-L-rhamnopyranose-(1-4)-beta-D-glucopyranuronic acid-(1-6)-[alpha-L-arabinofuranose-(1-3)][alpha-L-arabinofuranose-(1-4)]beta-D-galactopyranose-(1-6)-beta-D-galactopyranose
著者Cartmell, A, Gilbert, H.J.
登録日2017-10-30
公開日2018-10-17
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献A surface endogalactanase in Bacteroides thetaiotaomicron confers keystone status for arabinogalactan degradation.
Nat Microbiol, 3, 2018
6EUH
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BU of 6euh by Molmil
The GH43, Beta 1,3 Galactosidase, BT3683 with galactodeoxynojirimycin
分子名称: (2R,3S,4R,5S)-2-(hydroxymethyl)piperidine-3,4,5-triol, Beta-glucanase, CALCIUM ION
著者Cartmell, A, Gilbert, H.J.
登録日2017-10-30
公開日2018-10-17
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献A surface endogalactanase in Bacteroides thetaiotaomicron confers keystone status for arabinogalactan degradation.
Nat Microbiol, 3, 2018
6EUG
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BU of 6eug by Molmil
The GH43, Beta 1,3 Galactosidase, BT3683 with galactoimidazole
分子名称: Beta-glucanase, GLUCOIMIDAZOLE
著者Cartmell, A, Gilbert, H.J.
登録日2017-10-30
公開日2018-10-17
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.61 Å)
主引用文献A surface endogalactanase in Bacteroides thetaiotaomicron confers keystone status for arabinogalactan degradation.
Nat Microbiol, 3, 2018
8AA3
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BU of 8aa3 by Molmil
Core SusCD transporter units from the inactive levan utilisome in the presence of levan fructo-oligosaccharides DP 15-25
分子名称: MAGNESIUM ION, SusC homolog, SusD homolog, ...
著者White, J.B.R, Silale, A, Ranson, N.A, van den Berg, B.
登録日2022-06-29
公開日2023-06-07
最終更新日2023-06-21
実験手法ELECTRON MICROSCOPY (2.7 Å)
主引用文献Outer membrane utilisomes mediate glycan uptake in gut Bacteroidetes.
Nature, 618, 2023
8A9Y
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BU of 8a9y by Molmil
Substrate-free levan utilisation machinery (utilisome)
分子名称: DUF4960 domain-containing protein, Glycoside hydrolase family 32, MAGNESIUM ION, ...
著者White, J.B.R, Silale, A, Ranson, N.A, van den Berg, B.
登録日2022-06-29
公開日2023-06-07
最終更新日2024-07-24
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Outer membrane utilisomes mediate glycan uptake in gut Bacteroidetes.
Nature, 618, 2023
8AA4
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BU of 8aa4 by Molmil
SusC components of the dextran utilisation system (utilisome)
分子名称: SusC homolog
著者White, J.B.R, Silale, A, Ranson, N.A, van den Berg, B.
登録日2022-06-29
公開日2023-06-07
最終更新日2024-07-24
実験手法ELECTRON MICROSCOPY (3.1 Å)
主引用文献Outer membrane utilisomes mediate glycan uptake in gut Bacteroidetes.
Nature, 618, 2023
8AA1
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BU of 8aa1 by Molmil
Core SusCD transporter units from the levan utilisome with levan fructo-oligosaccharides DP 8-12
分子名称: MAGNESIUM ION, SusC homolog, SusD homolog, ...
著者White, J.B.R, Silale, A, Ranson, N.A, van den Berg, B.
登録日2022-06-29
公開日2023-06-07
最終更新日2023-06-21
実験手法ELECTRON MICROSCOPY (2.9 Å)
主引用文献Outer membrane utilisomes mediate glycan uptake in gut Bacteroidetes.
Nature, 618, 2023
8AA0
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BU of 8aa0 by Molmil
Levan utilisation machinery (utilisome) with levan fructo-oligosaccharides DP 8-12
分子名称: DUF4960 domain-containing protein, Glycoside hydrolase family 32, MAGNESIUM ION, ...
著者White, J.B.R, Silale, A, Ranson, N.A, van den Berg, B.
登録日2022-06-29
公開日2023-06-07
最終更新日2023-06-21
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Outer membrane utilisomes mediate glycan uptake in gut Bacteroidetes.
Nature, 618, 2023
8AA2
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BU of 8aa2 by Molmil
Inactive levan utilisation machinery (utilisome) in the presence of levan fructo-oligosaccharides DP 15-25
分子名称: DUF4960 domain-containing protein, Glycoside hydrolase family 32, MAGNESIUM ION, ...
著者White, J.B.R, Silale, A, Ranson, N.A, van den Berg, B.
登録日2022-06-29
公開日2023-06-07
最終更新日2023-06-21
実験手法ELECTRON MICROSCOPY (3.1 Å)
主引用文献Outer membrane utilisomes mediate glycan uptake in gut Bacteroidetes.
Nature, 618, 2023
7ZNR
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BU of 7znr by Molmil
Inactive D62N mutant of BT1760 Endo-acting levanase from Bacteroides thetaiotaomicron VPI-5482
分子名称: SULFATE ION, Sucrose-6-phosphate hydrolase, beta-D-fructofuranose-(2-6)-beta-D-fructofuranose, ...
著者Basle, A, Bolam, D.
登録日2022-04-21
公開日2023-06-21
最終更新日2024-06-19
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献Outer membrane utilisomes mediate glycan uptake in gut Bacteroidetes.
Nature, 618, 2023
7ZNS
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BU of 7zns by Molmil
Inactive D62N mutant of BT1760 Endo-acting levanase from Bacteroides thetaiotaomicron VPI-5482
分子名称: Glycoside hydrolase family 32, SULFATE ION, beta-D-fructofuranose-(2-6)-beta-D-fructofuranose, ...
著者Basle, A, Bolam, D.
登録日2022-04-21
公開日2023-06-21
最終更新日2024-06-19
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Outer membrane utilisomes mediate glycan uptake in gut Bacteroidetes.
Nature, 618, 2023
3PP1
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BU of 3pp1 by Molmil
Crystal Structure of the Human Mitogen-activated protein kinase kinase 1 (MEK 1) in complex with ligand and MgATP
分子名称: 3-[(2R)-2,3-dihydroxypropyl]-6-fluoro-5-[(2-fluoro-4-iodophenyl)amino]-8-methylpyrido[2,3-d]pyrimidine-4,7(3H,8H)-dione, ACETATE ION, ADENOSINE-5'-TRIPHOSPHATE, ...
著者Dougan, D.R.
登録日2010-11-23
公開日2011-02-23
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Discovery of TAK-733, a potent and selective MEK allosteric site inhibitor for the treatment of cancer.
Bioorg.Med.Chem.Lett., 21, 2011
3P23
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BU of 3p23 by Molmil
Crystal structure of the Human kinase and RNase domains in complex with ADP
分子名称: ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, SULFATE ION, ...
著者Ali, M.M.U, Pearl, L.H.
登録日2010-10-01
公開日2011-02-23
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structure of the Ire1 autophosphorylation complex and implications for the unfolded protein response.
Embo J., 30, 2011
4Z3V
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BU of 4z3v by Molmil
Fragment-Based Discovery of a Small Molecule Reversible Inhibitor of Bruton's Tyrosine Kinase
分子名称: 1,2-ETHANEDIOL, 4-amino-8-(5-methyl-1H-indazol-6-yl)cinnoline-3-carboxamide, IMIDAZOLE, ...
著者Dougan, D.R.
登録日2015-03-31
公開日2015-07-01
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Fragment-Based Discovery of a Small Molecule Inhibitor of Bruton's Tyrosine Kinase.
J.Med.Chem., 58, 2015
4ZLZ
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BU of 4zlz by Molmil
Crystal Structure of Bruton's Tyrosine Kinase in complex with a substituted Cinnoline
分子名称: 4-amino-8-(4-methylpyridin-3-yl)cinnoline-3-carboxamide, DIMETHYL SULFOXIDE, IMIDAZOLE, ...
著者Dougan, D.R.
登録日2015-05-01
公開日2015-07-01
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Fragment-Based Discovery of a Small Molecule Inhibitor of Bruton's Tyrosine Kinase.
J.Med.Chem., 58, 2015
3MBL
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BU of 3mbl by Molmil
Crystal Structure of the human mitogen-activated protein kinase kinase 1 (MEK 1) in complex with ligand and MgADP
分子名称: 5-acetyl-2-[(2-fluoro-4-iodophenyl)amino]-N-(2-hydroxyethoxy)-1-methyl-1H-pyrrole-3-carboxamide, ADENOSINE-5'-DIPHOSPHATE, Dual specificity mitogen-activated protein kinase kinase 1, ...
著者Dougan, D.R, Mol, C.D.
登録日2010-03-25
公開日2010-07-28
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structure-based design and synthesis of pyrrole derivatives as MEK inhibitors.
Bioorg.Med.Chem.Lett., 20, 2010
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