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IRAK4 in complex with inhibitor
分子名称:	Interleukin-1 receptor-associated kinase 4, N-[(2R)-2-fluoranyl-3-methyl-3-oxidanyl-butyl]-6-[(6-fluoranylpyrazolo[1,5-a]pyrimidin-5-yl)amino]-4-(propan-2-ylamino)pyridine-3-carboxamide, SULFATE ION
著者	Ghosh, K, Bose, S.
登録日	2020-02-12
公開日	2020-11-25
実験手法	X-RAY DIFFRACTION (2.19 Å)
主引用文献	Optimization of Nicotinamides as Potent and Selective IRAK4 Inhibitors with Efficacy in a Murine Model of Psoriasis. Acs Med.Chem.Lett., 11, 2020

CRYSTAL STRUCTURE OF RAR-RELATED ORPHAN RECEPTOR C (NHIS-RORGT(244-487)-L6-SRC1(6T78-692) IN COMPLEX WITH A TRICYCLIC SULFONE RORGT INVERSE AGONIST
分子名称:	Nuclear receptor ROR-gamma, trans-4-[(3aR,9bR)-8-cyano-9b-[(4-fluorophenyl)sulfonyl]-7-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)-1,2,3a,4,5,9b-hexahydro-3H-benzo[e]indole-3-carbonyl]cyclohexane-1-carboxylic acid
著者	Sack, J.S.
登録日	2020-08-18
公開日	2020-09-16
最終更新日	2023-10-18
実験手法	X-RAY DIFFRACTION (2.43 Å)
主引用文献	Tricyclic sulfones as potent, selective and efficacious ROR gamma t inverse agonists - Exploring C6 and C8 SAR using late-stage functionalization. Bioorg.Med.Chem.Lett., 30, 2020

Structure of the effector-binding domain of deoxyribonucleoside regulator DeoR from Bacillus subtilis
分子名称:	BICINE, Deoxyribonucleoside regulator
著者	Rezacova, P, Skerlova, J.
登録日	2014-02-10
公開日	2014-06-04
最終更新日	2023-09-20
実験手法	X-RAY DIFFRACTION (1.8 Å)
主引用文献	Structure of the effector-binding domain of deoxyribonucleoside regulator DeoR from Bacillus subtilis. Febs J., 281, 2014

Structure of the effector-binding domain of deoxyribonucleoside regulator DeoR from Bacillus subtilis in complex with deoxyribose-5-phosphate
分子名称:	CADMIUM ION, COBALT (II) ION, Deoxyribonucleoside regulator, ...
著者	Rezacova, P, Skerlova, J.
登録日	2014-02-10
公開日	2014-06-04
最終更新日	2023-09-20
実験手法	X-RAY DIFFRACTION (1.6 Å)
主引用文献	Structure of the effector-binding domain of deoxyribonucleoside regulator DeoR from Bacillus subtilis. Febs J., 281, 2014