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7YIZ
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BU of 7yiz by Molmil
Crystal structure of anti-mPEG h15-2b Fab W104Y mutant
分子名称: 15-2b W104Y heavy chain, 15-2b light chain, 2,5,8,11,14,17-HEXAOXANONADECAN-19-OL
著者Chang, C.Y, Nguyen, T.M.T, Li, Y.C, Su, Y.C.
登録日2022-07-18
公開日2023-08-02
最終更新日2025-02-12
実験手法X-RAY DIFFRACTION (2.42 Å)
主引用文献Engineering a High-Affinity Anti-Methoxy Poly(ethylene glycol) (mPEG) Antibody for Sensitive Immunosensing of mPEGylated Therapeutics and mPEG Molecules
Bioconjug.Chem., 33, 2022
5QTW
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FACTOR XIA IN COMPLEX WITH THE INHIBITOR methyl (2R,7S)-7-({(2E)-3-[5-chloro-2-(1H-tetrazol-1-yl)phenyl]prop-2-enoyl}amino)-14-[(methoxycarbonyl)amino]-2,3,4,5,6,7-hexahydro-1H-8,11-epimino-1,9-benzodiazacyclotridecine-2-carboxylate
分子名称: 1,2-ETHANEDIOL, Coagulation factor XI, SULFATE ION, ...
著者Sheriff, S.
登録日2019-11-13
公開日2020-01-29
最終更新日2024-10-23
実験手法X-RAY DIFFRACTION (2.12 Å)
主引用文献Orally bioavailable amine-linked macrocyclic inhibitors of factor XIa.
Bioorg.Med.Chem.Lett., 30, 2020
5QTV
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FACTOR XIA IN COMPLEX WITH THE INHIBITOR methyl [(2R,7S)-7-({(2E)-3-[5-chloro-2-(1H-tetrazol-1-yl)phenyl]prop-2-enoyl}amino)-2-(trifluoromethyl)-2,3,4,5,6,7-hexahydro-1H-8,11-epimino-1,9-benzodiazacyclotridecin-14-yl]carbamate
分子名称: 1,2-ETHANEDIOL, Coagulation factor XI, SULFATE ION, ...
著者Sheriff, S.
登録日2019-11-13
公開日2020-01-29
最終更新日2024-10-23
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Orally bioavailable amine-linked macrocyclic inhibitors of factor XIa.
Bioorg.Med.Chem.Lett., 30, 2020
5QTX
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BU of 5qtx by Molmil
FACTOR XIA IN COMPLEX WITH THE INHIBITOR ethyl (2R,7S)-7-({(2E)-3-[5-chloro-2-(1H-tetrazol-1-yl)phenyl]prop-2-enoyl}amino)-14-[(methoxycarbonyl)amino]-1,2,3,4,5,6,7,9-octahydro-11,8-(azeno)-1,9-benzodiazacyclotridecine-2-carboxylate
分子名称: 1,2-ETHANEDIOL, Coagulation factor XI, SULFATE ION, ...
著者Sheriff, S.
登録日2019-11-13
公開日2020-01-29
最終更新日2024-10-23
実験手法X-RAY DIFFRACTION (2.07 Å)
主引用文献Orally bioavailable amine-linked macrocyclic inhibitors of factor XIa.
Bioorg.Med.Chem.Lett., 30, 2020
5QTY
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BU of 5qty by Molmil
FACTOR XIA IN COMPLEX WITH THE INHIBITOR ethyl (2R,7S)-7-({(2E)-3-[5-chloro-2-(1H-tetrazol-1-yl)phenyl]prop-2-enoyl}amino)-15-[(methoxycarbonyl)amino]-2,3,4,5,6,7-hexahydro-1H-12,8-(metheno)-1,9-benzodiazacyclotetradecine-2-carboxylate
分子名称: 1,2-ETHANEDIOL, Coagulation factor XI, SULFATE ION, ...
著者Sheriff, S.
登録日2019-11-13
公開日2020-01-29
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (1.89 Å)
主引用文献Orally bioavailable amine-linked macrocyclic inhibitors of factor XIa.
Bioorg.Med.Chem.Lett., 30, 2020
8HE4
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BU of 8he4 by Molmil
The structure of chitin deacetylase Pst_13661 from Puccinia striiformis f. sp. tritici
分子名称: Chitin deacetylase, ZINC ION, ~{N}-oxidanylnaphthalene-1-carboxamide
著者Liu, L, Li, Y.C, Zhou, Y, Yang, Q.
登録日2022-11-07
公開日2023-05-31
最終更新日2024-10-23
実験手法X-RAY DIFFRACTION (1.93 Å)
主引用文献Inhibition of chitin deacetylases to attenuate plant fungal diseases.
Nat Commun, 14, 2023
8HE1
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BU of 8he1 by Molmil
The structure of chitin deacetylase Pst_13661 from Puccinia striiformis f. sp. tritici
分子名称: BENZHYDROXAMIC ACID, Chitin deacetylase, ZINC ION
著者Liu, L, Li, Y.C, Zhou, Y, Yang, Q.
登録日2022-11-07
公開日2023-05-31
最終更新日2024-11-06
実験手法X-RAY DIFFRACTION (1.61 Å)
主引用文献Inhibition of chitin deacetylases to attenuate plant fungal diseases.
Nat Commun, 14, 2023
8HE2
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The structure of chitin deacetylase Pst_13661 from Puccinia striiformis f. sp. tritici
分子名称: Chitin deacetylase, ZINC ION, tert-butyl N-[3-[[4-(oxidanylcarbamoyl)phenyl]methylamino]-3-oxidanylidene-propyl]carbamate
著者Liu, L, Li, Y.C, Zhou, Y, Yang, Q.
登録日2022-11-07
公開日2023-05-31
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (1.61 Å)
主引用文献Inhibition of chitin deacetylases to attenuate plant fungal diseases.
Nat Commun, 14, 2023
8HF9
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BU of 8hf9 by Molmil
The structure of chitin deacetylase Pst_13661 from Puccinia striiformis f. sp. tritici
分子名称: Chitin deacetylase, ZINC ION
著者Liu, L, Li, Y.C, Zhou, Y, Yang, Q.
登録日2022-11-10
公開日2023-05-31
最終更新日2024-10-09
実験手法X-RAY DIFFRACTION (1.96 Å)
主引用文献Inhibition of chitin deacetylases to attenuate plant fungal diseases.
Nat Commun, 14, 2023
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件を2025-07-09に公開中

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