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4E5A
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BU of 4e5a by Molmil
The W197A mutant of p38a MAP kinase
分子名称: Mitogen-activated protein kinase 14
著者Livnah, O, Tzarum, N, Eisenberg-Domovich, Y.
登録日2012-03-14
公開日2012-10-31
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.87 Å)
主引用文献Lipid Molecules Induce p38 alpha Activation via a Novel Molecular Switch.
J.Mol.Biol., 424, 2012
4E6C
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BU of 4e6c by Molmil
p38a-perifosine Complex
分子名称: (1,1-dimethylpiperidin-1-ium-4-yl) octadecyl hydrogen phosphate, Mitogen-activated protein kinase 14
著者Livnah, O, Tzarum, N, Eisenberg-Domovich, Y.
登録日2012-03-15
公開日2012-10-31
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.39 Å)
主引用文献Lipid Molecules Induce p38 alpha Activation via a Novel Molecular Switch.
J.Mol.Biol., 424, 2012
4E8A
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BU of 4e8a by Molmil
The crystal structure of p38a MAP kinase in complex with PIA24
分子名称: (1R,2S,3R,4S,6S)-6-(cyclohexylmethoxy)-2,3,4-trihydroxycyclohexyl (2R)-2-methoxy-3-(octadecyloxy)propyl hydrogen (S)-phosphate, Mitogen-activated protein kinase 14
著者Livnah, O, Tzarum, N, Eisenberg-Domovich, Y.
登録日2012-03-20
公開日2012-10-31
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Lipid Molecules Induce p38 alpha Activation via a Novel Molecular Switch.
J.Mol.Biol., 424, 2012
4E6A
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BU of 4e6a by Molmil
p38a-PIA23 complex
分子名称: (2S)-2-methoxy-3-(octadecyloxy)propyl (1R,2R,3R,4S,6S)-2,3,4-trihydroxy-6-(2-methylpropoxy)cyclohexyl hydrogen (S)-phosphate, Mitogen-activated protein kinase 14
著者Livnah, O, Tzarum, N, Eisenberg-Domovich, Y.
登録日2012-03-15
公開日2012-10-31
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.09 Å)
主引用文献Lipid Molecules Induce p38 alpha Activation via a Novel Molecular Switch.
J.Mol.Biol., 424, 2012
6R6E
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BU of 6r6e by Molmil
Crystal structure of di-phosphorylated human CLK1 in complex with 5-(6,7-dichloro-1-methyl-1H-indol-3-yl)pyrimidin-4-amine
分子名称: 5-[6,7-bis(chloranyl)-1-methyl-indol-3-yl]pyrimidin-4-amine, Dual specificity protein kinase CLK1
著者Livnah, O, Domovich, Y.
登録日2019-03-27
公開日2020-05-06
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Crystal structure of di-phosphorylated human CLK1 in complex with 5-(6,7-dichloro-1-methyl-1H-indol-3-yl)pyrimidin-4-amine
To Be Published
6R3D
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BU of 6r3d by Molmil
Crystal structure of di-phosphorylated human CLK1 in complex with 4-(6,7-dichloro-1H-indol-3-yl)pyrimidin-2-amine
分子名称: 4-[6,7-bis(chloranyl)-1~{H}-indol-3-yl]pyrimidin-2-amine, Dual specificity protein kinase CLK1
著者Livnah, O, Domovich, Y.
登録日2019-03-20
公開日2020-04-08
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Crystal structure of di-phosphorylated human CLK1 in complex with 4-(1-methyl-1H-indol-3-yl)pyrimidin-2-amine
To Be Published
6R6X
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BU of 6r6x by Molmil
Crystal structure of di-phosphorylated human CLK1 in complex with 5-(1-methyl-1H-indol-3-yl)pyrimidin-4-amine
分子名称: 5-(1-methylindol-3-yl)pyrimidin-4-amine, Dual specificity protein kinase CLK1
著者Livnah, O, Domovich, Y.
登録日2019-03-28
公開日2020-05-06
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Crystal structure of di-phosphorylated human CLK1 in complex with 5-(1-methyl-1H-indol-3-yl)pyrimidin-4-amine
To Be Published
6R8J
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BU of 6r8j by Molmil
Crystal structure of di-phosphorylated human CLK1 in complex with 4-(1-methyl-1H-indol-3-yl)pyrimidin-2-amine
分子名称: 4-(1-methylindol-3-yl)pyrimidin-2-amine, Dual specificity protein kinase CLK1
著者Livnah, O, Domovich, Y.
登録日2019-04-02
公開日2020-05-13
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Non-phosphorylated human CLK1 in complex with an indole inhibitor to 1.65 Ang
To Be Published
2FHN
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BU of 2fhn by Molmil
Avidin related protein AVR4 (C122S, K109I mutant) in complex with BNA
分子名称: 5-(2-OXO-HEXAHYDRO-THIENO[3,4-D]IMIDAZOL-6-YL)-PENTANOIC ACID (4-NITRO-PHENYL)-AMIDE, Avidin-related protein 4/5, FORMIC ACID
著者Livnah, O, Prizant, M.
登録日2005-12-26
公開日2006-03-21
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Factors dictating the pseudocatalytic efficiency of avidins
J.Mol.Biol., 358, 2006
2FHL
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BU of 2fhl by Molmil
avidin related protein (AVR4)-BNA complex
分子名称: 5-(2-OXO-HEXAHYDRO-THIENO[3,4-D]IMIDAZOL-6-YL)-PENTANOIC ACID (4-NITRO-PHENYL)-AMIDE, Avidin-related protein 4/5, FORMIC ACID
著者Livnah, O, Prizant, M.
登録日2005-12-26
公開日2006-03-21
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.05 Å)
主引用文献Factors dictating the pseudocatalytic efficiency of avidins
J.Mol.Biol., 358, 2006
1IJ8
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BU of 1ij8 by Molmil
CRYSTAL STRUCTURE OF LITE AVIDIN-BNI COMPLEX
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 5-(2-OXO-HEXAHYDRO-THIENO[3,4-D]IMIDAZOL-6-YL)-PENTANOIC ACID (4-NITRO-PHENYL)-AMIDE, AVIDIN
著者Livnah, O, Huberman, T.
登録日2001-04-25
公開日2001-09-12
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Chicken avidin exhibits pseudo-catalytic properties. Biochemical, structural, and electrostatic consequences.
J.Biol.Chem., 276, 2001
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件を2024-08-07に公開中

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