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Structure of DYRK1A in complex with compound 53
分子名称:	4-[2-methyl-3-(2-pyridin-2-yloxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine, DIMETHYL SULFOXIDE, Dual specificity tyrosine-phosphorylation-regulated kinase 1A, ...
著者	Dokurno, P, Surgenor, A.E, Kotschy, A.
登録日	2020-09-29
公開日	2021-05-26
最終更新日	2024-11-20
実験手法	X-RAY DIFFRACTION (2.1 Å)
主引用文献	Structure-Guided Discovery of Potent and Selective DYRK1A Inhibitors. J.Med.Chem., 64, 2021

Structure of DYRK1A in complex with compound 38
分子名称:	4-(2,3-dibutylimidazo[4,5-b]pyridin-5-yl)pyridine-2,6-diamine, CHLORIDE ION, Dual specificity tyrosine-phosphorylation-regulated kinase 1A
著者	Dokurno, P, Surgenor, A.E, Kotschy, A.
登録日	2020-09-29
公開日	2021-05-26
最終更新日	2024-10-09
実験手法	X-RAY DIFFRACTION (2.1 Å)
主引用文献	Structure-Guided Discovery of Potent and Selective DYRK1A Inhibitors. J.Med.Chem., 64, 2021

Structure of DYRK1A in complex with compound 28
分子名称:	1-[4-(1-benzofuran-5-yl)pyridin-2-yl]piperazine, CHLORIDE ION, Dual specificity tyrosine-phosphorylation-regulated kinase 1A
著者	Dokurno, P, Surgenor, A.E, Kotschy, A.
登録日	2020-09-28
公開日	2021-05-26
最終更新日	2024-11-20
実験手法	X-RAY DIFFRACTION (2.2 Å)
主引用文献	Structure-Guided Discovery of Potent and Selective DYRK1A Inhibitors. J.Med.Chem., 64, 2021

Structure of DYRK1A in complex with compound 46
分子名称:	4-[2-methyl-3-(2-phenoxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine, CHLORIDE ION, Dual specificity tyrosine-phosphorylation-regulated kinase 1A
著者	Dokurno, P, Surgenor, A.E, Kotschy, A.
登録日	2020-09-29
公開日	2021-05-26
最終更新日	2024-10-16
実験手法	X-RAY DIFFRACTION (2.8 Å)
主引用文献	Structure-Guided Discovery of Potent and Selective DYRK1A Inhibitors. J.Med.Chem., 64, 2021