5SBL
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5sbl by Molmil](/molmil-images/mine/5sbl) | CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z126932614 | 分子名称: | 1,2-ETHANEDIOL, 2-[(methylsulfonyl)methyl]-1H-benzimidazole, CD44 antigen, ... | 著者 | Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O. | 登録日 | 2021-09-14 | 公開日 | 2021-09-22 | 実験手法 | X-RAY DIFFRACTION (1.198 Å) | 主引用文献 | CD44 PanDDA analysis group deposition To Be Published
|
|
5SBK
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5sbk by Molmil](/molmil-images/mine/5sbk) | CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z1258992717 | 分子名称: | 1,2-ETHANEDIOL, CD44 antigen, DIMETHYL SULFOXIDE, ... | 著者 | Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O. | 登録日 | 2021-09-14 | 公開日 | 2021-09-22 | 実験手法 | X-RAY DIFFRACTION (1.23 Å) | 主引用文献 | CD44 PanDDA analysis group deposition To Be Published
|
|
5SBO
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5sbo by Molmil](/molmil-images/mine/5sbo) | CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z2856434878 | 分子名称: | 1,2-ETHANEDIOL, 4-[(3,4-dimethoxyphenyl)methyl]morpholine, CD44 antigen, ... | 著者 | Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O. | 登録日 | 2021-09-14 | 公開日 | 2021-09-22 | 実験手法 | X-RAY DIFFRACTION (1.274 Å) | 主引用文献 | CD44 PanDDA analysis group deposition To Be Published
|
|
5SBP
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5sbp by Molmil](/molmil-images/mine/5sbp) | CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z1229798311 | 分子名称: | 1,2-ETHANEDIOL, 2-acetamido-6-fluorobenzoic acid, CD44 antigen, ... | 著者 | Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O. | 登録日 | 2021-09-14 | 公開日 | 2021-09-22 | 実験手法 | X-RAY DIFFRACTION (1.275 Å) | 主引用文献 | CD44 PanDDA analysis group deposition To Be Published
|
|
5SBQ
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5sbq by Molmil](/molmil-images/mine/5sbq) | CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z44592329 | 分子名称: | CD44 antigen, DIMETHYL SULFOXIDE, N-phenyl-N'-pyridin-3-ylurea, ... | 著者 | Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O. | 登録日 | 2021-09-14 | 公開日 | 2021-09-22 | 実験手法 | X-RAY DIFFRACTION (0.988 Å) | 主引用文献 | CD44 PanDDA analysis group deposition To Be Published
|
|
5SBR
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5sbr by Molmil](/molmil-images/mine/5sbr) | CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z1259341012 | 分子名称: | (1R)-1-[4-(morpholin-4-yl)phenyl]ethan-1-amine, 1,2-ETHANEDIOL, CD44 antigen, ... | 著者 | Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O. | 登録日 | 2021-09-14 | 公開日 | 2021-09-22 | 実験手法 | X-RAY DIFFRACTION (1.286 Å) | 主引用文献 | CD44 PanDDA analysis group deposition To Be Published
|
|
5SBT
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5sbt by Molmil](/molmil-images/mine/5sbt) | CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z445856640 | 分子名称: | 1,2-ETHANEDIOL, CD44 antigen, DIMETHYL SULFOXIDE, ... | 著者 | Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O. | 登録日 | 2021-09-14 | 公開日 | 2021-09-22 | 実験手法 | X-RAY DIFFRACTION (1.16 Å) | 主引用文献 | CD44 PanDDA analysis group deposition To Be Published
|
|
5SBU
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5sbu by Molmil](/molmil-images/mine/5sbu) | CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z839988838 | 分子名称: | CD44 antigen, DIMETHYL SULFOXIDE, N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]cyclohexanamine, ... | 著者 | Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O. | 登録日 | 2021-09-14 | 公開日 | 2021-09-22 | 実験手法 | X-RAY DIFFRACTION (1.044 Å) | 主引用文献 | CD44 PanDDA analysis group deposition To Be Published
|
|
5SBS
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5sbs by Molmil](/molmil-images/mine/5sbs) | CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z340495298 | 分子名称: | 1,2-ETHANEDIOL, CD44 antigen, DIMETHYL SULFOXIDE, ... | 著者 | Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O. | 登録日 | 2021-09-14 | 公開日 | 2021-09-22 | 実験手法 | X-RAY DIFFRACTION (1.024 Å) | 主引用文献 | CD44 PanDDA analysis group deposition To Be Published
|
|
5SBX
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5sbx by Molmil](/molmil-images/mine/5sbx) | CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z53825479 | 分子名称: | 1,2-ETHANEDIOL, CD44 antigen, DI(HYDROXYETHYL)ETHER, ... | 著者 | Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O. | 登録日 | 2021-09-14 | 公開日 | 2021-09-22 | 実験手法 | X-RAY DIFFRACTION (1.051 Å) | 主引用文献 | CD44 PanDDA analysis group deposition To Be Published
|
|
5SBW
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5sbw by Molmil](/molmil-images/mine/5sbw) | CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z2856434874 | 分子名称: | 1,2-ETHANEDIOL, 1-{[4-(propan-2-yl)phenyl]methyl}piperidin-4-ol, CD44 antigen, ... | 著者 | Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O. | 登録日 | 2021-09-14 | 公開日 | 2021-09-22 | 実験手法 | X-RAY DIFFRACTION (1.148 Å) | 主引用文献 | CD44 PanDDA analysis group deposition To Be Published
|
|
5SBV
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5sbv by Molmil](/molmil-images/mine/5sbv) | CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z31721798 | 分子名称: | 1,2-ETHANEDIOL, 3-cyclohexyl-1-(morpholin-4-yl)propan-1-one, CD44 antigen, ... | 著者 | Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O. | 登録日 | 2021-09-14 | 公開日 | 2021-09-22 | 実験手法 | X-RAY DIFFRACTION (1.109 Å) | 主引用文献 | CD44 PanDDA analysis group deposition To Be Published
|
|
5SBY
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5sby by Molmil](/molmil-images/mine/5sby) | CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z1878656559 | 分子名称: | (1R,2R)-2,4,4-trimethyl-N-[(1H-pyrazol-3-yl)methyl]cyclopentan-1-amine, 1,2-ETHANEDIOL, CD44 antigen, ... | 著者 | Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O. | 登録日 | 2021-09-14 | 公開日 | 2021-09-22 | 実験手法 | X-RAY DIFFRACTION (1.217 Å) | 主引用文献 | CD44 PanDDA analysis group deposition To Be Published
|
|
5SBZ
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5sbz by Molmil](/molmil-images/mine/5sbz) | CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z768399682 | 分子名称: | 1,2-ETHANEDIOL, CD44 antigen, DIMETHYL SULFOXIDE, ... | 著者 | Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O. | 登録日 | 2021-09-14 | 公開日 | 2021-09-22 | 実験手法 | X-RAY DIFFRACTION (1.17 Å) | 主引用文献 | CD44 PanDDA analysis group deposition To Be Published
|
|
5SC0
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5sc0 by Molmil](/molmil-images/mine/5sc0) | CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z2856434899 | 分子名称: | 1,2-ETHANEDIOL, 1-[(thiophen-3-yl)methyl]piperidin-4-ol, CD44 antigen, ... | 著者 | Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O. | 登録日 | 2021-09-14 | 公開日 | 2021-09-22 | 実験手法 | X-RAY DIFFRACTION (1.192 Å) | 主引用文献 | CD44 PanDDA analysis group deposition To Be Published
|
|
5SC1
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5sc1 by Molmil](/molmil-images/mine/5sc1) | CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z431807512 | 分子名称: | 1,2-ETHANEDIOL, CD44 antigen, DIMETHYL SULFOXIDE, ... | 著者 | Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O. | 登録日 | 2021-09-14 | 公開日 | 2021-09-22 | 実験手法 | X-RAY DIFFRACTION (1.165 Å) | 主引用文献 | CD44 PanDDA analysis group deposition To Be Published
|
|
5SC2
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5sc2 by Molmil](/molmil-images/mine/5sc2) | CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z190780124 | 分子名称: | (3S)-N-[(1R)-1-cyclopropylethyl]-2-oxo-2,3-dihydropyridine-3-carboxamide, 1,2-ETHANEDIOL, CD44 antigen, ... | 著者 | Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O. | 登録日 | 2021-09-14 | 公開日 | 2021-09-22 | 実験手法 | X-RAY DIFFRACTION (1.208 Å) | 主引用文献 | CD44 PanDDA analysis group deposition To Be Published
|
|
5SC3
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5sc3 by Molmil](/molmil-images/mine/5sc3) | CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z422471910 | 分子名称: | 1,2-ETHANEDIOL, CD44 antigen, DIMETHYL SULFOXIDE, ... | 著者 | Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O. | 登録日 | 2021-09-14 | 公開日 | 2021-09-22 | 実験手法 | X-RAY DIFFRACTION (1.24 Å) | 主引用文献 | CD44 PanDDA analysis group deposition To Be Published
|
|
5SC4
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5sc4 by Molmil](/molmil-images/mine/5sc4) | CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z927412236 | 分子名称: | (2R)-2-amino-1-[(2S)-2-methylpiperidin-1-yl]propan-1-one, 1,2-ETHANEDIOL, CD44 antigen, ... | 著者 | Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O. | 登録日 | 2021-09-14 | 公開日 | 2021-09-22 | 実験手法 | X-RAY DIFFRACTION (1.165 Å) | 主引用文献 | CD44 PanDDA analysis group deposition To Be Published
|
|
5SC5
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5sc5 by Molmil](/molmil-images/mine/5sc5) | CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z56827661 | 分子名称: | 1,2-ETHANEDIOL, CD44 antigen, DIMETHYL SULFOXIDE, ... | 著者 | Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O. | 登録日 | 2021-09-14 | 公開日 | 2021-09-22 | 実験手法 | X-RAY DIFFRACTION (1.171 Å) | 主引用文献 | CD44 PanDDA analysis group deposition To Be Published
|
|
5SC6
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5sc6 by Molmil](/molmil-images/mine/5sc6) | CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with POB0019 | 分子名称: | 1,2-ETHANEDIOL, CD44 antigen, DIMETHYL SULFOXIDE, ... | 著者 | Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O. | 登録日 | 2021-09-14 | 公開日 | 2021-09-22 | 実験手法 | X-RAY DIFFRACTION (1.327 Å) | 主引用文献 | CD44 PanDDA analysis group deposition To Be Published
|
|
5SC7
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5sc7 by Molmil](/molmil-images/mine/5sc7) | CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with POB0120 | 分子名称: | (2R)-1',4'-dihydro-2'H-spiro[pyrrolidine-2,3'-quinolin]-2'-one, 1,2-ETHANEDIOL, CD44 antigen, ... | 著者 | Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O. | 登録日 | 2021-09-14 | 公開日 | 2021-09-22 | 実験手法 | X-RAY DIFFRACTION (1.197 Å) | 主引用文献 | CD44 PanDDA analysis group deposition To Be Published
|
|
5A3N
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5a3n by Molmil](/molmil-images/mine/5a3n) | Crystal structure of human PLU-1 (JARID1B) in complex with KDOAM25a | 分子名称: | 1,2-ETHANEDIOL, 2-[[[2-[2-(dimethylamino)ethyl-ethyl-amino]-2-oxidanylidene-ethyl]amino]methyl]pyridine-4-carboxamide, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, ... | 著者 | Srikannathasan, V, Johansson, C, Gileadi, C, Nuzzi, A, Ruda, G.F, Kopec, J, von Delft, F, Arrowsmith, C.H, Bountra, C, Edwards, A, Brennan, P, Oppermann, U. | 登録日 | 2015-06-02 | 公開日 | 2015-07-08 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Potent and Selective KDM5 Inhibitor Stops Cellular Demethylation of H3K4me3 at Transcription Start Sites and Proliferation of MM1S Myeloma Cells. Cell Chem Biol, 24, 2017
|
|
4UF0
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4uf0 by Molmil](/molmil-images/mine/4uf0) | Crystal structure of JmjC domain of human histone demethylase UTY in complex with epitherapuetic compound 2-(((2-((2-(dimethylamino)ethyl) (ethyl)amino)-2-oxoethyl)amino)methyl)isonicotinic acid. | 分子名称: | 1,2-ETHANEDIOL, 2-{[(2-{[(E)-2-(dimethylamino)ethenyl](ethyl)amino}-2-oxoethyl)amino]methyl}pyridine-4-carboxylic acid, FE (II) ION, ... | 著者 | Srikannathasan, V, Johansson, C, Gileadi, C, Tobias, K, Kopec, J, von Delft, F, Arrowsmith, C.H, Bountra, C, Edwards, A, Oppermann, U. | 登録日 | 2014-12-22 | 公開日 | 2015-01-14 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.78 Å) | 主引用文献 | Structural Analysis of Human Kdm5B Guides Histone Demethylase Inhibitor Development. Nat.Chem.Biol., 12, 2016
|
|
5A1F
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5a1f by Molmil](/molmil-images/mine/5a1f) | Crystal structure of the catalytic domain of PLU1 in complex with N-oxalylglycine. | 分子名称: | 1,2-ETHANEDIOL, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, LYSINE-SPECIFIC DEMETHYLASE 5B, ... | 著者 | Srikannathasan, V, Johansson, C, Strain-Damerell, C, Gileadi, C, Szykowska, A, Kupinska, K, Kopec, J, Krojer, T, Steuber, H, von Delft, F, Burgess-Brown, N.A, Arrowsmith, C.H, Bountra, C, Edwards, A.M, Oppermann, U. | 登録日 | 2015-04-29 | 公開日 | 2015-05-06 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structural Analysis of Human Kdm5B Guides Histone Demethylase Inhibitor Development. Nat.Chem.Biol., 12, 2016
|
|