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1GFW
THE 2.8 ANGSTROM CRYSTAL STRUCTURE OF CASPASE-3 (APOPAIN OR CPP32)IN COMPLEX WITH AN ISATIN SULFONAMIDE INHIBITOR.
Descriptor:
1-METHYL-5-(2-PHENOXYMETHYL-PYRROLIDINE-1-SULFONYL)-1H-INDOLE-2,3-DIONE, CASPASE-3 (APOPAIN, P10), ...
Authors:
Concha, N.O
,
Janson, C.A.
Deposit date:
2000-06-16
Release date:
2000-06-23
Last modified:
2024-11-13
Method:
X-RAY DIFFRACTION (2.8 Å)
Cite:
Potent and selective nonpeptide inhibitors of caspases 3 and 7 inhibit apoptosis and maintain cell functionality.
J.Biol.Chem., 275, 2000
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PDB entries from 2025-07-09