7FQR
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![BU of 7fqr by Molmil](/molmil-images/mine/7fqr) | PanDDA analysis group deposition -- Crystal structure of PTP1B in complex with FMOOA000666a | Descriptor: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1, methyl (1S,3S,4R)-4-hydroxy-3-[(1S)-1-hydroxypropyl]-2-azabicyclo[2.2.2]octane-2-carboxylate | Authors: | Mehlman, T, Biel, J, Azeem, S.M, Nelson, E.R, Hossain, S, Dunnett, L.E, Paterson, N.G, Douangamath, A, Talon, R, Axford, D, Orins, H, von Delft, F, Keedy, D.A. | Deposit date: | 2022-10-19 | Release date: | 2022-11-23 | Last modified: | 2024-05-22 | Method: | X-RAY DIFFRACTION (1.9 Å) | Cite: | Room-temperature crystallography reveals altered binding of small-molecule fragments to PTP1B. Elife, 12, 2023
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7FRE
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![BU of 7fre by Molmil](/molmil-images/mine/7fre) | PanDDA analysis group deposition -- Crystal structure of PTP1B after initial refinement with no ligand modeled | Descriptor: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1 | Authors: | Mehlman, T, Biel, J, Azeem, S.M, Nelson, E.R, Hossain, S, Dunnett, L.E, Paterson, N.G, Douangamath, A, Talon, R, Axford, D, Orins, H, von Delft, F, Keedy, D.A. | Deposit date: | 2022-10-20 | Release date: | 2022-11-23 | Last modified: | 2024-05-22 | Method: | X-RAY DIFFRACTION (1.85 Å) | Cite: | Room-temperature crystallography reveals altered binding of small-molecule fragments to PTP1B. Elife, 12, 2023
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7FRN
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![BU of 7frn by Molmil](/molmil-images/mine/7frn) | PanDDA analysis group deposition -- Crystal structure of PTP1B in complex with Z915492990 | Descriptor: | 1-methyl-N-[(thiophen-2-yl)methyl]-1H-pyrazole-5-carboxamide, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1 | Authors: | Mehlman, T, Biel, J, Azeem, S.M, Nelson, E.R, Hossain, S, Dunnett, L.E, Paterson, N.G, Douangamath, A, Talon, R, Axford, D, Orins, H, von Delft, F, Keedy, D.A. | Deposit date: | 2022-10-24 | Release date: | 2022-11-23 | Last modified: | 2024-05-22 | Method: | X-RAY DIFFRACTION (1.85 Å) | Cite: | Room-temperature crystallography reveals altered binding of small-molecule fragments to PTP1B. Elife, 12, 2023
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7GU4
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![BU of 7gu4 by Molmil](/molmil-images/mine/7gu4) | |
7GTY
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![BU of 7gty by Molmil](/molmil-images/mine/7gty) | |
7GU3
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![BU of 7gu3 by Molmil](/molmil-images/mine/7gu3) | |
7GU1
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![BU of 7gu1 by Molmil](/molmil-images/mine/7gu1) | |
7GU0
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![BU of 7gu0 by Molmil](/molmil-images/mine/7gu0) | |
7GU2
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![BU of 7gu2 by Molmil](/molmil-images/mine/7gu2) | |
7GU5
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![BU of 7gu5 by Molmil](/molmil-images/mine/7gu5) | |
7GU8
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![BU of 7gu8 by Molmil](/molmil-images/mine/7gu8) | |
7GU6
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![BU of 7gu6 by Molmil](/molmil-images/mine/7gu6) | |
7GUB
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![BU of 7gub by Molmil](/molmil-images/mine/7gub) | |
7GUA
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![BU of 7gua by Molmil](/molmil-images/mine/7gua) | |
7GUC
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![BU of 7guc by Molmil](/molmil-images/mine/7guc) | |
7GTZ
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![BU of 7gtz by Molmil](/molmil-images/mine/7gtz) | |
7GTX
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![BU of 7gtx by Molmil](/molmil-images/mine/7gtx) | |
7GU7
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![BU of 7gu7 by Molmil](/molmil-images/mine/7gu7) | |
7GTW
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![BU of 7gtw by Molmil](/molmil-images/mine/7gtw) | |
7GU9
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![BU of 7gu9 by Molmil](/molmil-images/mine/7gu9) | |
7GSJ
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![BU of 7gsj by Molmil](/molmil-images/mine/7gsj) | |
7GT1
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![BU of 7gt1 by Molmil](/molmil-images/mine/7gt1) | PanDDA Analysis group deposition -- Crystal structure of PTP1B in complex with FMOMB000209a | Descriptor: | (2S)-2-(2-chloro-6-fluorophenyl)-2,3-dihydroquinazolin-4(1H)-one, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1 | Authors: | Mehlman, T, Ginn, H.M, Keedy, D.A. | Deposit date: | 2024-01-03 | Release date: | 2024-01-24 | Last modified: | 2024-04-24 | Method: | X-RAY DIFFRACTION (1.91 Å) | Cite: | An expanded view of ligandability in the allosteric enzyme PTP1B from computational reanalysis of large-scale crystallographic data. Biorxiv, 2024
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7GSG
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![BU of 7gsg by Molmil](/molmil-images/mine/7gsg) | |
7GTI
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![BU of 7gti by Molmil](/molmil-images/mine/7gti) | PanDDA Analysis group deposition -- Crystal structure of PTP1B in complex with FMOOA000571a | Descriptor: | 1-{(1S,4R,5S,6R)-6-hydroxy-4-[(pyridin-2-yl)oxy]-2-azabicyclo[3.3.1]nonan-2-yl}ethan-1-one, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1 | Authors: | Mehlman, T, Ginn, H.M, Keedy, D.A. | Deposit date: | 2024-01-03 | Release date: | 2024-01-24 | Last modified: | 2024-04-24 | Method: | X-RAY DIFFRACTION (1.66 Å) | Cite: | An expanded view of ligandability in the allosteric enzyme PTP1B from computational reanalysis of large-scale crystallographic data. Biorxiv, 2024
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7GSB
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![BU of 7gsb by Molmil](/molmil-images/mine/7gsb) | |