9BHS
Crystal structure of the WDR domain of human DCAF1 in complex with OICR-9939 compound
This is a non-PDB format compatible entry.
Summary for 9BHS
Entry DOI | 10.2210/pdb9bhs/pdb |
Descriptor | DDB1- and CUL4-associated factor 1, (4P)-N-[(1S)-3-amino-1-(3-chloro-4-fluorophenyl)-3-oxopropyl]-4-(4-chloro-2-fluorophenyl)-5-(1-methyl-1H-pyrazol-4-yl)-1H-pyrrole-3-carboxamide, UNKNOWN LIGAND, ... (4 entities in total) |
Functional Keywords | wd-repeat, wdr, dcaf1, sgc, structural genomics, psi-2, protein structure initiative, structural genomics consortium, transferase |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 2 |
Total formula weight | 72312.65 |
Authors | kimani, S.,Dong, A.,Li, Y.,Seitova, A.,Al-Awar, R.,Wilson, B.,Ackloo, S.,Arrowsmith, C.H.,Edwards, A.M.,Halabelian, L.,Structural Genomics Consortium (SGC) (deposition date: 2024-04-21, release date: 2024-05-01) |
Primary citation | kimani, S.,Dong, A.,Li, Y.,Seitova, A.,Al-Awar, R.,Wilson, B.,Ackloo, S.,Arrowsmith, C.H.,Edwards, A.M.,Halabelian, L. Crystal structure of the WDR domain of human DCAF1 in complex with OICR-9939 compound To be published, |
Experimental method | X-RAY DIFFRACTION (1.43 Å) |
Structure validation
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