9BRK
Crystal Structure of Human G Protein-Coupled Receptor Kinase 5 in Complex with GRL098-22
This is a non-PDB format compatible entry.
Summary for 9BRK
| Entry DOI | 10.2210/pdb9brk/pdb |
| Descriptor | G protein-coupled receptor kinase 5, tert-butyl (3R)-3-({5-[(Z)-(5-{[(1R)-1-(4-fluorophenyl)ethyl]carbamoyl}-2-oxo-1,2-dihydro-3H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrol-3-yl}carbamoyl)piperazine-1-carboxylate (3 entities in total) |
| Functional Keywords | g protein-coupled receptor, gpcr g protein-coupled receptor kinase, grk kinase, signaling protein-inhibitor complex, signaling protein/inhibitor |
| Biological source | Homo sapiens (human) |
| Total number of polymer chains | 1 |
| Total formula weight | 69562.44 |
| Authors | |
| Primary citation | Chen, Y.,Tesmer, J.J.G. Structures of GRK5 bound to novel inhibitors To Be Published, |
| Experimental method | X-RAY DIFFRACTION (2.7 Å) |
Structure validation
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