Summary for 8VOF
Entry DOI | 10.2210/pdb8vof/pdb |
Descriptor | Isoform 2 of Phosphatidylinositol 4-kinase beta,Isoform 2 of Phosphatidylinositol 4-kinase beta,Phosphatidylinositol 4-kinase beta, Ras-related protein Rab-11A, methyl 2-chloro-5-(methyl{(8R)-3-[4-(methylcarbamoyl)phenyl]pyrazolo[1,5-a]pyridine-5-carbonyl}amino)benzoate, ... (6 entities in total) |
Functional Keywords | inhibitor complex, chimera, cryptosporidiosis, transferase |
Biological source | Homo sapiens (human) More |
Total number of polymer chains | 2 |
Total formula weight | 86225.64 |
Authors | Knapp, M.S.,Cuellar, C.,Mamo, M. (deposition date: 2024-01-15, release date: 2024-09-04, Last modification date: 2024-09-25) |
Primary citation | Manjunatha, U.H.,Diagana, T.T. Cryptosporidium PI(4)K inhibitor EDI048 is a gut-restricted parasiticidal agent to treat paediatric enteric cryptosporidiosis Nat Microbiol, 2024 |
Experimental method | X-RAY DIFFRACTION (3 Å) |
Structure validation
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