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8VOF

GI targeted CpPI4K inhibitor

This is a non-PDB format compatible entry.
Summary for 8VOF
Entry DOI10.2210/pdb8vof/pdb
DescriptorIsoform 2 of Phosphatidylinositol 4-kinase beta,Isoform 2 of Phosphatidylinositol 4-kinase beta,Phosphatidylinositol 4-kinase beta, Ras-related protein Rab-11A, methyl 2-chloro-5-(methyl{(8R)-3-[4-(methylcarbamoyl)phenyl]pyrazolo[1,5-a]pyridine-5-carbonyl}amino)benzoate, ... (6 entities in total)
Functional Keywordsinhibitor complex, chimera, cryptosporidiosis, transferase
Biological sourceHomo sapiens (human)
More
Total number of polymer chains2
Total formula weight86225.64
Authors
Knapp, M.S.,Cuellar, C.,Mamo, M. (deposition date: 2024-01-15, release date: 2024-09-04)
Primary citationManjunatha, U.H.,Diagana, T.T.
Rational design of GI targeted parasiticidal agent to treat pediatric enteric cryptosporidiosis
To Be Published,
Experimental method
X-RAY DIFFRACTION (3 Å)
Structure validation

224572

건을2024-09-04부터공개중

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