8V2T
Phosphoheptose isomerase GMHA from Burkholderia pseudomallei bound to inhibitor Mut148591
Summary for 8V2T
Entry DOI | 10.2210/pdb8v2t/pdb |
Related | 8V4J |
Descriptor | Phosphoheptose isomerase, 1,5,6-trideoxy-6,6-difluoro-1-(N-hydroxyformamido)-6-phosphono-D-ribo-hexitol, ZINC ION, ... (6 entities in total) |
Functional Keywords | heptose biosynthesis, isomerase-inhibitor complex, isomerase/inhibitor |
Biological source | Burkholderia pseudomallei 1106a |
Total number of polymer chains | 1 |
Total formula weight | 23826.51 |
Authors | Junop, M.S.,Brown, C.,Szabla, R. (deposition date: 2023-11-23, release date: 2023-12-06, Last modification date: 2024-05-01) |
Primary citation | Moreau, F.,Atamanyuk, D.,Blaukopf, M.,Barath, M.,Herczeg, M.,Xavier, N.M.,Monbrun, J.,Airiau, E.,Henryon, V.,Leroy, F.,Floquet, S.,Bonnard, D.,Szabla, R.,Brown, C.,Junop, M.S.,Kosma, P.,Gerusz, V. Potentiating Activity of GmhA Inhibitors on Gram-Negative Bacteria. J.Med.Chem., 67:6610-6623, 2024 Cited by PubMed: 38598312DOI: 10.1021/acs.jmedchem.4c00037 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.402 Å) |
Structure validation
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