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8TYF

Plasmodium vivax PMV-WM06 inhibitor complex

This is a non-PDB format compatible entry.
Summary for 8TYF
Entry DOI10.2210/pdb8tyf/pdb
DescriptorPlasmepsin V, 2-acetamido-2-deoxy-beta-D-glucopyranose, (2E,4aR,7aS)-6-[(3M)-3-(2-chlorophenyl)pyridin-2-yl]-7a-(2,5-difluorophenyl)-2-imino-3-methyloctahydro-4H-pyrrolo[3,4-d]pyrimidin-4-one, ... (5 entities in total)
Functional Keywordsplasmepsinix, plasmepsinx, inhibitor, hydrolase, hydrolase-inhibitor complex, hydrolase/inhibitor
Biological sourcePlasmodium vivax Sal-1
Total number of polymer chains1
Total formula weight53654.91
Authors
Hodder, A.N.,Scally, S.W.,Czabotar, P.E.,Cowman, A.F. (deposition date: 2023-08-25, release date: 2024-08-28)
Primary citationHodder, A.N.,Cowman, A.F.,Scally, S.W.
Plasmodium vivax PMX-XX inhibitor complex
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.59 Å)
Structure validation

224572

건을2024-09-04부터공개중

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