8SX2
PARP4 catalytic domain bound to EB47
Summary for 8SX2
Entry DOI | 10.2210/pdb8sx2/pdb |
Descriptor | Protein mono-ADP-ribosyltransferase PARP4, 2-[4-[(2S,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]carbonylpiperazin-1-yl]-N-(1-oxidanylidene-2,3-dihydroisoindol-4-yl)ethanamide (3 entities in total) |
Functional Keywords | parp family, adp-ribosyltransferase, marylation, vault, transferase |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 2 |
Total formula weight | 75594.77 |
Authors | Frigon, L.,Pascal, J.M. (deposition date: 2023-05-19, release date: 2023-11-08, Last modification date: 2023-12-20) |
Primary citation | Frigon, L.,Pascal, J.M. Structural and biochemical analysis of the PARP1-homology region of PARP4/vault PARP. Nucleic Acids Res., 51:12492-12507, 2023 Cited by PubMed: 37971310DOI: 10.1093/nar/gkad1064 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.95 Å) |
Structure validation
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