8SC8
Structure of PI3KG in complex with MTX-531
Summary for 8SC8
Entry DOI | 10.2210/pdb8sc8/pdb |
Descriptor | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform, SULFATE ION, N-[(5P)-2-chloro-5-(4-{[(1R)-1-phenylethyl]amino}quinazolin-6-yl)pyridin-3-yl]methanesulfonamide, ... (4 entities in total) |
Functional Keywords | pi3kg, dual egfr/pi3k inhibitor, transferase, transferase-inhibitor complex, transferase/inhibitor |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 1 |
Total formula weight | 111661.36 |
Authors | |
Primary citation | Whitehead, C.E.,Leopold, J. Structure of PI3KG in complex with MTX-531 To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.687 Å) |
Structure validation
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