8R4U
Structure of salt-inducible kinase 3 with inhibitors
Summary for 8R4U
Entry DOI | 10.2210/pdb8r4u/pdb |
Descriptor | Serine/threonine-protein kinase SIK3, scFvH1, 8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(3-fluoranylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one, ... (5 entities in total) |
Functional Keywords | kinase, inhibitor complex, drug design, ampk-like kinase, uba, ligase |
Biological source | Homo sapiens (human) More |
Total number of polymer chains | 8 |
Total formula weight | 263571.46 |
Authors | |
Primary citation | Oster, L.,Castaldo, M.,de Vries, E.,Edfeldt, F.,Pemberton, N.,Gordon, E.,Cederblad, L.,Kack, H. The structures of salt-inducible kinase 3 in complex with inhibitors reveal determinants for binding and selectivity. J.Biol.Chem., 300:107201-107201, 2024 Cited by PubMed: 38508313DOI: 10.1016/j.jbc.2024.107201 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.416 Å) |
Structure validation
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