8QWY
Crystal structure of human Casein Kinase II subunit alpha (CK2a1) in complex with 4-(6-((5-isopropoxy-2-methoxyphenyl)amino)pyrazin-2-yl)benzoic acid
Summary for 8QWY
Entry DOI | 10.2210/pdb8qwy/pdb |
Descriptor | Casein kinase II subunit alpha, SULFATE ION, 4-[6-[(2-methoxy-5-propan-2-yloxy-phenyl)amino]pyrazin-2-yl]benzoic acid, ... (4 entities in total) |
Functional Keywords | ck2, inhibitor, kinase, transferase |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 2 |
Total formula weight | 82567.53 |
Authors | Kraemer, A.,Galal, K.,Willson, T.,Knapp, S.,Structural Genomics Consortium (SGC) (deposition date: 2023-10-20, release date: 2024-01-17) |
Primary citation | Kraemer, A.,Galal, K.,Willson, T.,Knapp, S.,Structural Genomics Consortium (SGC) Crystal structure of human Casein Kinase II subunit alpha (CK2a1) in complex with 4-(6-(6-isopropoxy-1H-indol-1-yl)pyrazin-2-yl)benzoic acid To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.6 Å) |
Structure validation
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