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8P9X

Vitamin D receptor complex with Xe4Me agonist ligand

Summary for 8P9X
Entry DOI10.2210/pdb8p9x/pdb
DescriptorVitamin D3 receptor A, Nuclear receptor coactivator 2, ACETATE ION, ... (5 entities in total)
Functional Keywordsnuclear receptor, agonist, ligand binding domain, transcription
Biological sourceDanio rerio (zebrafish)
More
Total number of polymer chains2
Total formula weight36108.15
Authors
Rochel, N. (deposition date: 2023-06-06, release date: 2024-06-26, Last modification date: 2024-07-24)
Primary citationLen-Tayon, K.,Beraud, C.,Fauveau, C.,Belorusova, A.Y.,Chebaro, Y.,Mourino, A.,Massfelder, T.,Chauchereau, A.,Metzger, D.,Rochel, N.,Laverny, G.
A vitamin D-based strategy overcomes chemoresistance in prostate cancer.
Br.J.Pharmacol., 2024
Cited by
PubMed: 38982588
DOI: 10.1111/bph.16492
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.15 Å)
Structure validation

223532

數據於2024-08-07公開中

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