8JUD
Crystal structure of human MMP-7 in complex with inhibitor
Summary for 8JUD
Entry DOI | 10.2210/pdb8jud/pdb |
Descriptor | Matrilysin, Peptide Inhibitor, CALCIUM ION, ... (5 entities in total) |
Functional Keywords | matrilysin, matrin, matrix metalloproteinase-7, pump-1 protease, uterine metalloproteinase, hydrolase, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor |
Biological source | Homo sapiens (human) More |
Total number of polymer chains | 2 |
Total formula weight | 20337.95 |
Authors | Kamitani, M.,Abe-Sato, K.,Oka, Y. (deposition date: 2023-06-26, release date: 2023-11-01, Last modification date: 2023-11-22) |
Primary citation | Abe-Sato, K.,Tabuse, H.,Kanazawa, H.,Kamitani, M.,Endo, M.,Tokura, S.,Wakabayashi, S.,Yahara, T.,Takeda, T.,Hitaka, K.,Gunji, E.,Kojima, N.,Oka, Y. Structure-Based Optimization and Biological Evaluation of Potent and Selective MMP-7 Inhibitors for Kidney Fibrosis. J.Med.Chem., 66:14653-14668, 2023 Cited by PubMed: 37861435DOI: 10.1021/acs.jmedchem.3c01166 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.5 Å) |
Structure validation
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