8JOF
solution-structure of Ras Binding Domain (RBD) in C-RAF
Summary for 8JOF
Entry DOI | 10.2210/pdb8jof/pdb |
Descriptor | RAF proto-oncogene serine/threonine-protein kinase (1 entity in total) |
Functional Keywords | mapk, signaling protein |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 1 |
Total formula weight | 9615.22 |
Authors | Makino, Y.,Matsumoto, S.,Yoshikawa, Y.,Kawamura, T.,Kumasaka, T.,Shima, F. (deposition date: 2023-06-07, release date: 2024-06-12) |
Primary citation | Yoshikawa, Y.,Makino, Y.,Hirokazu, K.,Kawamura, T.,Matsumoto, S.,Yuki, H.,Shibaike, A.,Okamura, M.,Okada, T.,Kataoka, T.,Honma, T.,Kumasaka, T.,Koyama, H.,Shima, F. Small-molecule RAS/RAF-binding Inhibitors Allosterically Disrupt RAF Conformation and Exert Efficacy Against Broad-spectrum RAS-driven Cancers To Be Published, |
Experimental method | SOLUTION NMR |
Structure validation
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