8JNZ
Human ADP-ribosyltransferase 1 (PARP1) catalytic domain bound to a pyrazolopyrimidine carboxamide inhibitor
Summary for 8JNZ
Entry DOI | 10.2210/pdb8jnz/pdb |
Descriptor | Poly [ADP-ribose] polymerase 1, processed C-terminus, 6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide, SULFATE ION (3 entities in total) |
Functional Keywords | dna adp-ribosyltransferase 1, parp1, parp inhibitor, transferase |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 2 |
Total formula weight | 79943.21 |
Authors | |
Primary citation | Wang, X.Y.,Wang, C.Y.,Zhou, J.,Xu, B.L. Human ADP-ribosyltransferase 1 (PARP1) catalytic domain bound to a pyrazolopyrimidine carboxamide inhibitor To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.84 Å) |
Structure validation
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