8I5M
Rat Kir4.1 in complex with PIP2
Summary for 8I5M
Entry DOI | 10.2210/pdb8i5m/pdb |
EMDB information | 35195 |
Descriptor | ATP-sensitive inward rectifier potassium channel 10, [(2R)-2-octanoyloxy-3-[oxidanyl-[(1R,2R,3S,4R,5R,6S)-2,3,6-tris(oxidanyl)-4,5-diphosphonooxy-cyclohexyl]oxy-phosphoryl]oxy-propyl] octanoate (2 entities in total) |
Functional Keywords | kir4.1, ion channel, transport protein, membrane protein |
Biological source | Rattus norvegicus (Norway rat) |
Total number of polymer chains | 4 |
Total formula weight | 158153.16 |
Authors | |
Primary citation | Zhou, X.,Zhao, C.,Xu, H.,Xu, Y.,Zhan, L.,Wang, P.,He, J.,Lu, T.,Gu, Y.,Yang, Y.,Xu, C.,Chen, Y.,Liu, Y.,Zeng, Y.,Tian, F.,Chen, Q.,Xie, X.,Liu, J.,Hu, H.,Li, J.,Zheng, Y.,Guo, J.,Gao, Z. Pharmacological inhibition of Kir4.1 evokes rapid-onset antidepressant responses. Nat.Chem.Biol., 20:857-866, 2024 Cited by PubMed: 38355723DOI: 10.1038/s41589-024-01555-y PDB entries with the same primary citation |
Experimental method | ELECTRON MICROSCOPY (2.85 Å) |
Structure validation
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