8FRZ
Full-length mouse 5-HT3A receptor in complex with serotonin, pre-activated
Summary for 8FRZ
Entry DOI | 10.2210/pdb8frz/pdb |
EMDB information | 29409 29410 29411 29418 |
Descriptor | 5-hydroxytryptamine receptor 3A, SEROTONIN, 2-acetamido-2-deoxy-beta-D-glucopyranose (3 entities in total) |
Functional Keywords | partial agonist, cys-loop, plgic, ion channel, transport protein |
Biological source | Mus musculus (house mouse) |
Total number of polymer chains | 5 |
Total formula weight | 315948.26 |
Authors | Felt, K.C.,Chakrapani, S. (deposition date: 2023-01-09, release date: 2023-12-27, Last modification date: 2024-05-01) |
Primary citation | Felt, K.,Stauffer, M.,Salas-Estrada, L.,Guzzo, P.R.,Xie, D.,Huang, J.,Filizola, M.,Chakrapani, S. Structural basis for partial agonism in 5-HT 3A receptors. Nat.Struct.Mol.Biol., 31:598-609, 2024 Cited by PubMed: 38177669DOI: 10.1038/s41594-023-01140-2 PDB entries with the same primary citation |
Experimental method | ELECTRON MICROSCOPY (2.75 Å) |
Structure validation
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