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8F4Q

rat branched chain ketoacid dehydrogenase kinase in complex with inhibtors

Summary for 8F4Q
Entry DOI10.2210/pdb8f4q/pdb
Descriptor[3-methyl-2-oxobutanoate dehydrogenase [lipoamide]] kinase, mitochondrial, ADENOSINE-5'-DIPHOSPHATE, SULFATE ION, ... (5 entities in total)
Functional Keywordsbranched chain ketoacid dehydrogenase kinase, inhibitor, signaling protein, transferase-inhibitor complex, transferase/inhibitor
Biological sourceRattus
Total number of polymer chains1
Total formula weight45590.92
Authors
Liu, S. (deposition date: 2022-11-11, release date: 2023-12-13)
Primary citationRoth Flach, R.,Filipski, K.,Bollinger, E.
Discovery of branched-chain ketoacid dehydrogenase kinase (BDK) inhibitors acting as stabilizers or destabilizers
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.151 Å)
Structure validation

221051

数据于2024-06-12公开中

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