8F4Q
rat branched chain ketoacid dehydrogenase kinase in complex with inhibtors
Summary for 8F4Q
Entry DOI | 10.2210/pdb8f4q/pdb |
Descriptor | [3-methyl-2-oxobutanoate dehydrogenase [lipoamide]] kinase, mitochondrial, ADENOSINE-5'-DIPHOSPHATE, SULFATE ION, ... (5 entities in total) |
Functional Keywords | branched chain ketoacid dehydrogenase kinase, inhibitor, signaling protein, transferase-inhibitor complex, transferase/inhibitor |
Biological source | Rattus |
Total number of polymer chains | 1 |
Total formula weight | 45590.92 |
Authors | |
Primary citation | Roth Flach, R.,Filipski, K.,Bollinger, E. Discovery of branched-chain ketoacid dehydrogenase kinase (BDK) inhibitors acting as stabilizers or destabilizers To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.151 Å) |
Structure validation
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