8F1W
EGFR(T790M/V948R) kinase in complex with poziotinib
Summary for 8F1W
Entry DOI | 10.2210/pdb8f1w/pdb |
Descriptor | Epidermal growth factor receptor, 1-[4-[4-[[3,4-bis(chloranyl)-2-fluoranyl-phenyl]amino]-7-methoxy-quinazolin-6-yl]oxypiperidin-1-yl]propan-1-one (2 entities in total) |
Functional Keywords | egfr, kinase, inhibitor, transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 4 |
Total formula weight | 152871.82 |
Authors | |
Primary citation | Beyett, T.S.,Eck, M.J. EGFR(T790M/V948R) kinase in complex with poziotinib To be published, |
Experimental method | X-RAY DIFFRACTION (3.2 Å) |
Structure validation
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