8F1H
EGFR kinase in complex with TAS6417 (CLN-081)
Summary for 8F1H
Entry DOI | 10.2210/pdb8f1h/pdb |
Descriptor | Epidermal growth factor receptor, N-[(5P,8S,10R)-4-amino-6-methyl-5-(quinolin-3-yl)-8,9-dihydropyrimido[5,4-b]indolizin-8-yl]prop-2-enamide, CITRIC ACID, ... (4 entities in total) |
Functional Keywords | egfr, kinase, exon 20, inhibitor, transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 1 |
Total formula weight | 38225.01 |
Authors | |
Primary citation | Beyett, T.S.,Eck, M.J. EGFR kinase in complex with TAS6417 (CLN-081) To be published, |
Experimental method | X-RAY DIFFRACTION (2.8 Å) |
Structure validation
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