8BD9
Crystal structure of TRIM33 alpha PHD-Bromo domain in complex with 10
Summary for 8BD9
Entry DOI | 10.2210/pdb8bd9/pdb |
Related | 8BD8 |
Descriptor | E3 ubiquitin-protein ligase TRIM33, 1,3-dimethylbenzimidazol-2-one, ZINC ION, ... (5 entities in total) |
Functional Keywords | trim33 alpha, phd-bromo domain, complex, transcription |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 1 |
Total formula weight | 24402.66 |
Authors | Tassone, G.,Pozzi, C.,Palomba, T. (deposition date: 2022-10-18, release date: 2022-12-07, Last modification date: 2024-01-31) |
Primary citation | Palomba, T.,Tassone, G.,Vacca, C.,Bartalucci, M.,Valeri, A.,Pozzi, C.,Cross, S.,Siragusa, L.,Desantis, J. Exploiting ELIOT for Scaffold-Repurposing Opportunities: TRIM33 a Possible Novel E3 Ligase to Expand the Toolbox for PROTAC Design. Int J Mol Sci, 23:-, 2022 Cited by PubMed: 36430693DOI: 10.3390/ijms232214218 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (3.2 Å) |
Structure validation
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