8P22
X-ray structure of acetylcholine-binding protein (AChBP) in complex with IOTA376.
Summary for 8P22
Entry DOI | 10.2210/pdb8p22/pdb |
Descriptor | Acetylcholine-binding protein, 2-[(2~{R})-1-ethylimidazolidin-2-yl]-6-pyridin-2-yl-pyridine, SULFATE ION, ... (5 entities in total) |
Functional Keywords | fragment based drug design, acetylcholine-binding protein, choline-binding proteins, choline-binding protein |
Biological source | Lymnaea stagnalis (great pond snail) |
Total number of polymer chains | 10 |
Total formula weight | 237209.54 |
Authors | Cederfelt, D.,Boronat, P.,Dobritzsch, D.,Hennig, S.,Fitzgerald, E.A.,de Esch, I.J.P.,Danielson, U.H. (deposition date: 2023-05-14, release date: 2024-05-08) |
Primary citation | Fitzgerald, E.A.,Cederfelt, D.,Boronat, P.,Aarmo Lund, B.,Dobritzsch, D.,de Esch, I.J.P.,Danielson, U.H. Elucidating the regulation of ligand gated ion channels via biophysical studies of ligand-induced conformational dynamics of acetylcholine binding proteins To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.2 Å) |
Structure validation
Download full validation report