8K5X
Crystal structure of human proMMP-9 catalytic domain in complex with inhibitor
Summary for 8K5X
Entry DOI | 10.2210/pdb8k5x/pdb |
Descriptor | Matrix metalloproteinase-9, ZINC ION, CALCIUM ION, ... (7 entities in total) |
Functional Keywords | mmp-9, 92 kda gelatinase, 92 kda type iv collagenase, gelatinase b, hydrolase |
Biological source | Homo sapiens (human) More |
Total number of polymer chains | 2 |
Total formula weight | 55648.40 |
Authors | |
Primary citation | Nishikawa-Shimono, R.,Kuwabara, M.,Fujisaki, S.,Matsuda, D.,Endo, M.,Kamitani, M.,Futamura, A.,Nomura, Y.,Yamaguchi-Sasaki, T.,Yabuuchi, T.,Yamaguchi, C.,Tanaka-Yamamoto, N.,Satake, S.,Abe-Sato, K.,Funayama, K.,Sakata, M.,Takahashi, S.,Hirano, K.,Fukunaga, T.,Uozumi, Y.,Kato, S.,Tamura, Y.,Nakamori, T.,Mima, M.,Mishima-Tsumagari, C.,Nozawa, D.,Imai, Y.,Asami, T. Discovery of novel indole derivatives as potent and selective inhibitors of proMMP-9 activation. Bioorg.Med.Chem.Lett., 97:129541-129541, 2023 Cited by PubMed: 37952596DOI: 10.1016/j.bmcl.2023.129541 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.9 Å) |
Structure validation
Download full validation report