8EGQ
Branched chain ketoacid dehydrogenase kinase complexes
Summary for 8EGQ
Entry DOI | 10.2210/pdb8egq/pdb |
Related | 8EGD 8EGF |
Descriptor | [3-methyl-2-oxobutanoate dehydrogenase [lipoamide]] kinase, mitochondrial, ADENOSINE-5'-DIPHOSPHATE, (2S)-2-ethyl-4-{[(2'M)-2'-(1H-tetrazol-5-yl)[1,1'-biphenyl]-4-yl]methyl}-3,4-dihydro-2H-pyrido[3,2-b][1,4]oxazine, ... (5 entities in total) |
Functional Keywords | branched-chain ketoacid dehydrogenase, branched-chain ketoacid dehydrogenase kinase, inhibitors, angiotensin receptor blocker, signaling protein, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Rattus norvegicus (Rat) |
Total number of polymer chains | 1 |
Total formula weight | 45581.77 |
Authors | |
Primary citation | Liu, S.,Kormos, B.L.,Knafels, J.D.,Sahasrabudhe, P.V.,Rosado, A.,Sommese, R.F.,Reyes, A.R.,Ward, J.,Roth Flach, R.J.,Wang, X.,Buzon, L.M.,Reese, M.R.,Bhattacharya, S.K.,Omoto, K.,Filipski, K.J. Structural studies identify angiotensin II receptor blocker-like compounds as branched-chain ketoacid dehydrogenase kinase inhibitors. J.Biol.Chem., 299:102959-102959, 2023 Cited by PubMed: 36717078DOI: 10.1016/j.jbc.2023.102959 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.955 Å) |
Structure validation
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