7ZEH
Human cytosolic 5' nucleotidase IIIB in complex with 3,4-diF-Bn7Guanine
Summary for 7ZEH
Entry DOI | 10.2210/pdb7zeh/pdb |
Descriptor | 7-methylguanosine phosphate-specific 5'-nucleotidase, N7-(3,4-difluorobenzyl) guanine, D-ribulose, ... (8 entities in total) |
Functional Keywords | cytosolic 5' nucleotidase, n7 methylguanosine monophosphate dephosphorylation, mrna cap degradation, hydrolase |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 4 |
Total formula weight | 143077.54 |
Authors | Kubacka, D.,Kozarski, M.,Baranowski, M.R.,Wojcik, R.,Jemielity, J.,Kowalska, J.,Basquin, J. (deposition date: 2022-03-31, release date: 2022-05-25, Last modification date: 2024-01-31) |
Primary citation | Kubacka, D.,Kozarski, M.,Baranowski, M.R.,Wojcik, R.,Panecka-Hofman, J.,Strzelecka, D.,Basquin, J.,Jemielity, J.,Kowalska, J. Substrate-Based Design of Cytosolic Nucleotidase IIIB Inhibitors and Structural Insights into Inhibition Mechanism. Pharmaceuticals, 15:-, 2022 Cited by PubMed: 35631380DOI: 10.3390/ph15050554 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.5 Å) |
Structure validation
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