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7ZEG

Human cytosolic 5' nucleotidase IIIB in complex with 3,4-diF-Bn7GMP

Summary for 7ZEG
Entry DOI10.2210/pdb7zeg/pdb
Descriptor7-methylguanosine phosphate-specific 5'-nucleotidase, N7-(3,4-difluorobenzyl) guanosine 5'-monophosphate, 1,2-ETHANEDIOL, ... (5 entities in total)
Functional Keywordscytosolic 5' nucleotidase, n7 methylguanosine monophosphate dephosphorylation, mrna cap degradation, hydrolase
Biological sourceHomo sapiens (human)
Total number of polymer chains2
Total formula weight70690.98
Authors
Kubacka, D.,Kozarski, M.,Baranowski, M.R.,Wojcik, R.,Jemielity, J.,Kowalska, J.,Basquin, J. (deposition date: 2022-03-31, release date: 2022-04-13, Last modification date: 2024-01-31)
Primary citationKubacka, D.,Kozarski, M.,Baranowski, M.R.,Wojcik, R.,Panecka-Hofman, J.,Strzelecka, D.,Basquin, J.,Jemielity, J.,Kowalska, J.
Substrate-Based Design of Cytosolic Nucleotidase IIIB Inhibitors and Structural Insights into Inhibition Mechanism.
Pharmaceuticals, 15:-, 2022
Cited by
PubMed: 35631380
DOI: 10.3390/ph15050554
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.56 Å)
Structure validation

221051

數據於2024-06-12公開中

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