7U22
Mycobacterium tuberculosis RNA polymerase sigma A holoenzyme open promoter complex containing UMN-7
Summary for 7U22
Entry DOI | 10.2210/pdb7u22/pdb |
Descriptor | DNA-directed RNA polymerase subunit alpha, MAGNESIUM ION, DNA-directed RNA polymerase subunit beta, ... (10 entities in total) |
Functional Keywords | transcription, inhibitor, rifabutin, transcription initiation, tuberculosis, mtb, mycobacterium tuberculosis, mycobacterium smegmatis, antibiotic |
Biological source | Mycobacterium tuberculosis More |
Total number of polymer chains | 8 |
Total formula weight | 435378.85 |
Authors | Molodtsov, V.,Ebright, R.H. (deposition date: 2022-02-22, release date: 2022-10-19, Last modification date: 2023-10-18) |
Primary citation | Lan, T.,Ganapathy, U.S.,Sharma, S.,Ahn, Y.M.,Zimmerman, M.,Molodtsov, V.,Hegde, P.,Gengenbacher, M.,Ebright, R.H.,Dartois, V.,Freundlich, J.S.,Dick, T.,Aldrich, C.C. Redesign of Rifamycin Antibiotics to Overcome ADP-Ribosylation-Mediated Resistance. Angew.Chem.Int.Ed.Engl., 61:e202211498-e202211498, 2022 Cited by PubMed: 36222275DOI: 10.1002/anie.202211498 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (3.87 Å) |
Structure validation
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