7T9H
HIV Integrase in complex with Compound-15
7T9H の概要
エントリーDOI | 10.2210/pdb7t9h/pdb |
分子名称 | Integrase, MAGNESIUM ION, (2S)-tert-butoxy[2-methyl-4-(4-methylphenyl)quinolin-3-yl]acetic acid, ... (4 entities in total) |
機能のキーワード | dna integration, aids, rnaseh, ledgf, endonuclease, hiv-1 integrase, dna binding protein, viral protein |
由来する生物種 | Human immunodeficiency virus 1 |
タンパク質・核酸の鎖数 | 2 |
化学式量合計 | 37018.71 |
構造登録者 | |
主引用文献 | Naidu, B.N.,Patel, M.,McAuliffe, B.,Ding, B.,Cianci, C.,Simmermacher, J.,Jenkins, S.,Parker, D.D.,Sivaprakasam, P.,Khan, J.A.,Kish, K.,Lewis, H.,Hanumegowda, U.,Krystal, M.,Meanwell, N.A.,Kadow, J.F. Design, Synthesis, and Preclinical Profiling of GSK3739936 (BMS-986180), an Allosteric Inhibitor of HIV-1 Integrase with Broad-Spectrum Activity toward 124/125 Polymorphs. J.Med.Chem., 65:4949-4971, 2022 Cited by PubMed: 35235334DOI: 10.1021/acs.jmedchem.1c02169 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (2.53 Å) |
構造検証レポート
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