7PX6
PARP15 catalytic domain in complex with OUL241
Summary for 7PX6
Entry DOI | 10.2210/pdb7px6/pdb |
Related | 7PW3 7PWA 7PWC 7PWK 7PWL 7PWM 7PWP 7PWQ 7PWR 7PWS 7PWU 7PWW |
Descriptor | Protein mono-ADP-ribosyltransferase PARP15, 6-[(2-fluorophenyl)methoxy]phthalazine-1,4-dione, (4S)-2-METHYL-2,4-PENTANEDIOL, ... (4 entities in total) |
Functional Keywords | adp-ribosyltransferase, inhibitor, complex, transferase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 2 |
Total formula weight | 51281.33 |
Authors | Maksimainen, M.M.,Lehtio, L. (deposition date: 2021-10-08, release date: 2022-05-11, Last modification date: 2024-01-31) |
Primary citation | Nizi, M.G.,Maksimainen, M.M.,Murthy, S.,Massari, S.,Alaviuhkola, J.,Lippok, B.E.,Sowa, S.T.,Galera-Prat, A.,Prunskaite-Hyyrylainen, R.,Luscher, B.,Korn, P.,Lehtio, L.,Tabarrini, O. Potent 2,3-dihydrophthalazine-1,4-dione derivatives as dual inhibitors for mono-ADP-ribosyltransferases PARP10 and PARP15. Eur.J.Med.Chem., 237:114362-114362, 2022 Cited by PubMed: 35500474DOI: 10.1016/j.ejmech.2022.114362 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.65 Å) |
Structure validation
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