Summary for 7PA3
Entry DOI | 10.2210/pdb7pa3/pdb |
Descriptor | Parkinson disease protein 7, (3~{S})-~{N}-[5-[2-[(azanylidene-$l^{4}-azanylidene)amino]ethanoyl]-6,7-dihydro-4~{H}-[1,3]thiazolo[5,4-c]pyridin-2-yl]-1-(iminomethyl)pyrrolidine-3-carboxamide (3 entities in total) |
Functional Keywords | deglycase, inhibitor, unknown function |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 20495.72 |
Authors | Kim, R.Q.,Jia, Y.,Sapmaz, A.,Geurink, P.P. (deposition date: 2021-07-28, release date: 2022-08-10, Last modification date: 2024-01-31) |
Primary citation | Jia, Y.,Kim, R.Q.,Kooij, R.,Ovaa, H.,Sapmaz, A.,Geurink, P.P. Chemical Toolkit for PARK7: Potent, Selective, and High-Throughput. J.Med.Chem., 65:13288-13304, 2022 Cited by PubMed: 36149939DOI: 10.1021/acs.jmedchem.2c01113 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.42 Å) |
Structure validation
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