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7OPG

Crystal structure of CLK1 in complex with compound 2 (CC513)

Summary for 7OPG
Entry DOI10.2210/pdb7opg/pdb
DescriptorDual specificity protein kinase CLK1, 4-[2-(propylamino)imidazo[2,1-b][1,3,4]thiadiazol-5-yl]phenol, GLYCEROL, ... (6 entities in total)
Functional Keywordskinase inhibitor, clk1, splicing kinase, structural genomics, structural genomics consortium, sgc, transferase
Biological sourceHomo sapiens (Human)
Total number of polymer chains3
Total formula weight120916.75
Authors
Chaikuad, A.,Routier, S.,Bonnet, P.,Knapp, S.,Structural Genomics Consortium (SGC) (deposition date: 2021-05-31, release date: 2021-07-21, Last modification date: 2024-01-31)
Primary citationChaikuad, A.,Routier, S.,Bonnet, P.,Knapp, S.,Structural Genomics Consortium (SGC)
Crystal structure of CLK1 in complex with compound 2 (CC513)
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.93 Å)
Structure validation

221716

건을2024-06-26부터공개중

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