7MYH
Ubiquitin variant UbV.k.2 in complex with Ube2k
Summary for 7MYH
Entry DOI | 10.2210/pdb7myh/pdb |
Descriptor | Ubiquitin-conjugating enzyme E2 K, Ubiquitin variant UbV.k.2, GLYCEROL, ... (4 entities in total) |
Functional Keywords | ubiquitin conjugating enzyme, degradation, ubiquitin variant, inhibitor, transferase-inhibitor complex, transferase/inhibitor |
Biological source | Homo sapiens (Human) More |
Total number of polymer chains | 2 |
Total formula weight | 33055.57 |
Authors | Middleton, A.J.,Day, C.L.,Teyra, J.,Sidhu, S.S. (deposition date: 2021-05-21, release date: 2021-08-25, Last modification date: 2023-10-18) |
Primary citation | Middleton, A.J.,Teyra, J.,Zhu, J.,Sidhu, S.S.,Day, C.L. Identification of Ubiquitin Variants That Inhibit the E2 Ubiquitin Conjugating Enzyme, Ube2k. Acs Chem.Biol., 16:1745-1756, 2021 Cited by PubMed: 34397214DOI: 10.1021/acschembio.1c00445 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.394 Å) |
Structure validation
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