Summary for 7M0T
Entry DOI | 10.2210/pdb7m0t/pdb |
Descriptor | Dual specificity mitogen-activated protein kinase kinase 1, Serine/threonine-protein kinase B-raf, 5-[(4-bromo-2-chlorophenyl)amino]-4-fluoro-N-(2-hydroxyethoxy)-1-methyl-1H-benzimidazole-6-carboxamide, ... (5 entities in total) |
Functional Keywords | braf, mek1, transferase |
Biological source | Homo sapiens (Human) More |
Total number of polymer chains | 2 |
Total formula weight | 77407.07 |
Authors | Li, K.,Gonzalez Del-Pino, G.,Ha, B.H.,Park, E.,Eck, M.J. (deposition date: 2021-03-11, release date: 2021-04-21, Last modification date: 2023-10-18) |
Primary citation | Gonzalez-Del Pino, G.L.,Li, K.,Park, E.,Schmoker, A.M.,Ha, B.H.,Eck, M.J. Allosteric MEK inhibitors act on BRAF/MEK complexes to block MEK activation. Proc.Natl.Acad.Sci.USA, 118:-, 2021 Cited by PubMed: 34470822DOI: 10.1073/pnas.2107207118 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (3.19 Å) |
Structure validation
Download full validation report