7LEL
Crystal structure of the second bromodomain (BD2) of human BRDT bound to Bromosporine
Summary for 7LEL
Entry DOI | 10.2210/pdb7lel/pdb |
Descriptor | Bromodomain testis-specific protein, Bromosporine (3 entities in total) |
Functional Keywords | brdt, bet, plk1, testis specific, bromodomain, gene regulation |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 4 |
Total formula weight | 56436.94 |
Authors | Chan, A.,Karim, M.R.,Schonbrunn, E. (deposition date: 2021-01-14, release date: 2021-07-14, Last modification date: 2023-10-18) |
Primary citation | Karim, R.M.,Bikowitz, M.J.,Chan, A.,Zhu, J.Y.,Grassie, D.,Becker, A.,Berndt, N.,Gunawan, S.,Lawrence, N.J.,Schonbrunn, E. Differential BET Bromodomain Inhibition by Dihydropteridinone and Pyrimidodiazepinone Kinase Inhibitors. J.Med.Chem., 64:15772-15786, 2021 Cited by PubMed: 34710325DOI: 10.1021/acs.jmedchem.1c01096 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.15 Å) |
Structure validation
Download full validation report