7KYF
Botulism Neurooxin Light Chain A app form
Summary for 7KYF
Entry DOI | 10.2210/pdb7kyf/pdb |
Descriptor | Bont/A1, ZINC ION, N-[(3,5-dichlorophenyl)sulfonyl]-L-isoleucyl-N-hydroxy-L-norvalinamide, ... (4 entities in total) |
Functional Keywords | bont, botulinum neurotoxin nva-ila dipetpide bound, toxin |
Biological source | Clostridium botulinum |
Total number of polymer chains | 1 |
Total formula weight | 48296.82 |
Authors | Ortega, M.E.,Salzameda, N.T. (deposition date: 2020-12-07, release date: 2021-04-14, Last modification date: 2023-10-18) |
Primary citation | Amezcua, M.,Cruz, R.S.,Ku, A.,Moran, W.,Ortega, M.E.,Salzameda, N.T. Discovery of Dipeptides as Potent Botulinum Neurotoxin A Light-Chain Inhibitors. Acs Med.Chem.Lett., 12:295-301, 2021 Cited by PubMed: 33603978DOI: 10.1021/acsmedchemlett.0c00674 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.33 Å) |
Structure validation
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