7F7G
a linear Peptide Inhibitors in complex with GK domain
Summary for 7F7G
Entry DOI | 10.2210/pdb7f7g/pdb |
Descriptor | DLG4 GK domain, UNK-ARG-ILE-ARG-ARG-ASP-GLU-TYR-LEU-LYS-ALA-ILE-GLN-UNK (3 entities in total) |
Functional Keywords | maguk dlg stapled peptide linear peptide, peptide binding protein |
Biological source | Rattus norvegicus (Rat) More |
Total number of polymer chains | 4 |
Total formula weight | 46588.57 |
Authors | |
Primary citation | Unarta, I.C.,Xu, J.,Shang, Y.,Cheung, C.H.P.,Zhu, R.,Chen, X.,Cao, S.,Cheung, P.P.,Bierer, D.,Zhang, M.,Huang, X.,Li, X. Entropy of stapled peptide inhibitors in free state is the major contributor to the improvement of binding affinity with the GK domain. Rsc Chem Biol, 2:1274-1284, 2021 Cited by PubMed: 34458841DOI: 10.1039/d1cb00087j PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.446 Å) |
Structure validation
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