7EJV
The co-crystal structure of DYRK2 with YK-2-69
Summary for 7EJV
Entry DOI | 10.2210/pdb7ejv/pdb |
Descriptor | Dual specificity tyrosine-phosphorylation-regulated kinase 2, [6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanone, ... (4 entities in total) |
Functional Keywords | phosphorylase kinase, transferase |
Biological source | Homo sapiens (human) More |
Total number of polymer chains | 2 |
Total formula weight | 90842.83 |
Authors | |
Primary citation | Yuan, K.,Li, Z.,Kuang, W.,Wang, X.,Ji, M.,Chen, W.,Ding, J.,Li, J.,Min, W.,Sun, C.,Ye, X.,Lu, M.,Wang, L.,Ge, H.,Jiang, Y.,Hao, H.,Xiao, Y.,Yang, P. Targeting dual-specificity tyrosine phosphorylation-regulated kinase 2 with a highly selective inhibitor for the treatment of prostate cancer. Nat Commun, 13:2903-2903, 2022 Cited by PubMed: 35614066DOI: 10.1038/s41467-022-30581-4 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.5 Å) |
Structure validation
Download full validation report