7B9R
Cys-45-tethered stabilizer 4 of 14-3-3(sigma)/ERa PPI
Summary for 7B9R
Entry DOI | 10.2210/pdb7b9r/pdb |
Descriptor | 14-3-3 protein sigma, Estrogen receptor, MAGNESIUM ION, ... (5 entities in total) |
Functional Keywords | protein-protein interaction; stabilization; hub protein; transcription factor, signaling protein |
Biological source | Homo sapiens (Human) More |
Total number of polymer chains | 2 |
Total formula weight | 27793.54 |
Authors | Sijbesma, E.,Ottmann, C. (deposition date: 2020-12-14, release date: 2021-07-07, Last modification date: 2024-01-31) |
Primary citation | Sijbesma, E.,Hallenbeck, K.K.,Andrei, S.A.,Rust, R.R.,Adriaans, J.M.C.,Brunsveld, L.,Arkin, M.R.,Ottmann, C. Exploration of a 14-3-3 PPI Pocket by Covalent Fragments as Stabilizers. Acs Med.Chem.Lett., 12:976-982, 2021 Cited by PubMed: 34136078DOI: 10.1021/acsmedchemlett.1c00088 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.15 Å) |
Structure validation
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