7B0T
Crystal structure of MLLT1 YEATS domain T3 mutant in complex with benzimidazole-amide based compound 1
Summary for 7B0T
Entry DOI | 10.2210/pdb7b0t/pdb |
Descriptor | Protein ENL, 3-iodanyl-4-methyl-~{N}-[2-(piperidin-1-ylmethyl)-3~{H}-benzimidazol-5-yl]benzamide, 1,2-ETHANEDIOL, ... (4 entities in total) |
Functional Keywords | t3 mutant, structural genomics, structural genomics consortium, sgc, transcription |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 18830.53 |
Authors | Ni, X.,Chaikuad, A.,Brennan, P.E.,Knapp, S.,Structural Genomics Consortium (SGC) (deposition date: 2020-11-21, release date: 2021-02-17, Last modification date: 2024-01-31) |
Primary citation | Ni, X.,Londregan, A.T.,Owen, D.R.,Knapp, S.,Chaikuad, A. Structure and Inhibitor Binding Characterization of Oncogenic MLLT1 Mutants. Acs Chem.Biol., 16:571-578, 2021 Cited by PubMed: 33749253DOI: 10.1021/acschembio.0c00960 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.05 Å) |
Structure validation
Download full validation report