7TTE
Tubulin-RB3_SLD in complex with compound 12j
Summary for 7TTE
Entry DOI | 10.2210/pdb7tte/pdb |
Descriptor | Tubulin alpha-1B chain, Tubulin beta chain, Stathmin-4, ... (9 entities in total) |
Functional Keywords | microtubule inhibitor, colchicine, cell cycle, cancer, inhibitor complex, cell cycle-inhibitor complex, cell cycle/inhibitor |
Biological source | Rattus norvegicus (Norway rat) More |
Total number of polymer chains | 5 |
Total formula weight | 214832.77 |
Authors | White, S.W.,Yun, M. (deposition date: 2022-02-01, release date: 2023-04-12, Last modification date: 2023-10-25) |
Primary citation | Pochampally, S.,Hartman, K.L.,Wang, R.,Wang, J.,Yun, M.K.,Parmar, K.,Park, H.,Meibohm, B.,White, S.W.,Li, W.,Miller, D.D. Design, Synthesis, and Biological Evaluation of Pyrimidine Dihydroquinoxalinone Derivatives as Tubulin Colchicine Site-Binding Agents That Displayed Potent Anticancer Activity Both In Vitro and In Vivo. Acs Pharmacol Transl Sci, 6:526-545, 2023 Cited by PubMed: 37082747DOI: 10.1021/acsptsci.2c00108 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.7 Å) |
Structure validation
Download full validation report